SCHEMBL11060122

SCHEMBL11060122

COC(=O)C(CCn1c(C(=O)c2cccc(OC)c2)ccc1S(C)(=O)=O)C(=O)OC

nearest known ligand 0.43

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.43
STS P08842 3/20 0.42
TAS1R3 Q7RTX0 1/20 0.40
TAS1R1 Q7RTX1 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
VNN1 O95497 2/20 0.39
CES2 O00748 1/20 0.39
CES1 P23141 1/20 0.39
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
HSD11B1 P28845 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11060469 0.87 ALDH1A1 (0.38) ALDH1A1L3MBTL1NPSR1
SCHEMBL11064901 0.82 TAS1R3 (0.41) ALDH1A1STSTAS1R3TAS1R1L3MBTL1
SCHEMBL11059125 0.82 EPHX2 (0.36)
SCHEMBL11060324 0.81 HTT (0.37) L3MBTL1
SCHEMBL11058804 0.79 ELANE (0.32) ALDH1A1NPSR1CES2CES1HSD11B1
SCHEMBL11060436 0.78 MAPT (0.36) ALDH1A1L3MBTL1NPSR1CYP2C9CYP2C19
SCHEMBL11057977 0.78 HPGD (0.42) ALDH1A1L3MBTL1CYP2C9
SCHEMBL11064181 0.76 DAO (0.35)
SCHEMBL11057980 0.76 TSHR (0.43) ALDH1A1L3MBTL1NPSR1
SCHEMBL11060953 0.75 HPGD (0.33) ALDH1A1NPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4458081-A ANTIINFLAMMATORY, ANALGESIC, ANTICOAGULANT, MUSCLE RELAXANT SYNTEX (U.S.A.) INC. (US) 1984-07-03 US disclosed
US-4454326-A 5-Aroyl 6-chloro or 6-bromo 1,2-dihydro-3H-pyrrolo[1,2-a]pyrrole-1,1-di-carboxylates SYNTEX (U.S.A.) INC. (US) 1984-06-12 US disclosed
US-4347187-A Process for preparing 5-aroyl 1,2-dihydro-3H-pyrrolo[1,2-a]pyrrole-1-carboxylic acids and novel intermediates therein SYNTEX (U.S.A.) INC. (US) 1982-08-31 US disclosed
US-4347186-A Process for preparing 5-aroyl 1,2-dihydro-3-H pyrrolo[1,2-a]pyrrole-1-carboxylic acids and novel intermediates therein SYNTEX (U.S.A.) INC. (US) 1982-08-31 US disclosed