SCHEMBL11063447

SCHEMBL11063447

C=CCOc1ccc(F)c2c1CCN(C)CC2

nearest known ligand 0.71

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRA2A P08913 4/20 0.71
ADRA2B P18089 4/20 0.71
ADRA2C P18825 4/20 0.71
ADRA1D P25100 1/20 0.50
ADRA1A P35348 1/20 0.50
ADRA1B P35368 1/20 0.50
HTR2C P28335 8/20 0.43
HTR2B P41595 5/20 0.43
HTR1A P08908 3/20 0.38
HTR2A P28223 5/20 0.36
SLC6A4 P31645 2/20 0.35
ADRB2 P07550 1/20 0.35
CHRM5 P08912 1/20 0.35
DRD2 P14416 1/20 0.35
DRD4 P21917 1/20 0.35
HRH2 P25021 1/20 0.35
HTR7 P34969 1/20 0.35
DRD3 P35462 1/20 0.35
HTR6 P50406 1/20 0.35
KCNH2 Q12809 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10349589 0.83 ADRA2A (0.72) ADRA2AADRA2BADRA2CADRA1DADRA1A
SCHEMBL11070770 0.83 ADRA2A (0.71) ADRA2AADRA2BADRA2CADRA1DADRA1A
SCHEMBL10349233 0.83 ADRA2A (1.00) ADRA2AADRA2BADRA2CADRA1DADRA1A
Hydrochloric Acid SCHEMBL10349227 0.82 ADRA2A (0.97) ADRA2AADRA2BADRA2CADRA1DADRA1A
SCHEMBL11069747 0.78 ADRA2A (1.00) ADRA2AADRA2BADRA2CADRA1DADRA1A
Hydrochloric Acid SCHEMBL11067993 0.77 ADRA2A (0.97) ADRA2AADRA2BADRA2CADRA1DADRA1A
SCHEMBL10349592 0.72 ADRA2A (0.40) ADRA2AADRA2BADRA2CADRA1DADRA1A
SCHEMBL3292980 0.69 ADRA2A (0.52) ADRA2AADRA2BADRA2CHTR2CHTR2B
SCHEMBL14236454 0.67 HTR2C (0.50) ADRA2AADRA2BADRA2CHTR2CHTR2B
SCHEMBL3440774 0.67 MAOA (0.43) ADRA2AADRA2BADRA2CADRA1DADRA1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4469634-A Allyloxy- and allylthio-2,3,4,5-tetrahydro-1H-3-benzazepines SMITHKLINE BECKMAN CORPORATION (US) 1984-09-04 US disclosed
EP-0103961-A1 Allyloxy- and allylthio-2,3,4,5-tetrahydro-1H-3-benzazepines SMITHKLINE BECKMAN CORPORATION (US) 1984-03-28 EP disclosed