SCHEMBL11064084

SCHEMBL11064084

CCOC(=O)C(=O)Nc1cccc(F)c1

nearest known ligand 0.68

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MAPT P10636 3/20 0.68
MEN1 O00255 2/20 0.57
KMT2A Q03164 2/20 0.57
GPR35 Q9HC97 1/20 0.54
HTT P42858 1/20 0.53
ALDH1A1 P00352 2/20 0.52
KDM4E B2RXH2 1/20 0.52
GAA P10253 1/20 0.52
TDP1 Q9NUW8 1/20 0.52
PTPN1 P18031 1/20 0.51
SMN1; SMN2 Q16637 1/20 0.51
POLB P06746 1/20 0.50
L3MBTL1 Q9Y468 1/20 0.49
CYP19A1 P11511 2/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11402843 0.89 MAPT (0.63) MAPTGPR35ALDH1A1GAAPOLB
SCHEMBL11453702 0.84 MAPT (0.58) MAPTMEN1KMT2AGPR35ALDH1A1
SCHEMBL11744132 0.84 MAPK1 (0.66) MAPTMEN1KMT2AHTTALDH1A1
SCHEMBL11064502 0.84 MEN1 (0.59) MAPTMEN1KMT2AKDM4EGAA
SCHEMBL10650215 0.82 MAPT (0.55) MAPTGPR35HTTALDH1A1GAA
SCHEMBL11612418 0.82 GPR35 (0.61) MAPTMEN1KMT2AGPR35HTT
SCHEMBL11651728 0.82 HPGD (0.61) MAPTMEN1KMT2AGPR35ALDH1A1
SCHEMBL11595669 0.82 ALDH1A1 (0.57) MAPTGPR35ALDH1A1GAASMN1; SMN2
SCHEMBL11065326 0.82 MAPT (0.55) MAPTGPR35ALDH1A1GAAPOLB
SCHEMBL3344883 0.82 CYP19A1 (0.64) MAPTGPR35ALDH1A1GAASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4483707-A PLANT SAFTENING AGENTS CIBA-GEIGY CORPORATION (US) 1984-11-20 US disclosed
US-4191840-A Oxamic acid derivatives AMERICAN HOME PRODUCTS CORPORATION (US) 1980-03-04 US disclosed
US-4160100-A OXAMIC ACID DERIVATIVES AMERICAN HOME PRODUCTS CORPORATION (US) 1979-07-03 US disclosed
US-4154961-A Oxamic acid derivatives AMERICAN HOME PRODUCTS CORPORATION (US) 1979-05-15 US disclosed
US-4137325-A Antisecretory oxamic acid esters AMERICAN HOME PRODUCTS CORPORATION (US) 1979-01-30 US disclosed
US-4069343-A OXAMIC ACID DERIVATIVES FOR THE PREVENTION OF IMMEDIATE TYPE HYPERSENSITIVITY REACTIONS AMERICAN HOME PRODUCTS CORPORATION (US) 1978-01-17 US disclosed
US-4054661-A Pyridyl oxamic acid derivatives and use in the prevention of allergic reactions AMERICAN HOME PRODUCTS CORPORATION (US) 1977-10-18 US disclosed
US-4054657-A Pyrimidinyl oxamic acids and esters, and compositions and methods for the suppression of allergic manifestations AMERICAN HOME PRODUCTS CORPORATION (US) 1977-10-18 US disclosed
US-4054666-A Compositions and methods of treating immediate hypersensitivity reactions with thiazolyl oxamic acid derivatives AMERICAN HOME PRODUCTS CORPORATION (US) 1977-10-18 US disclosed
US-4036837-A 2 Alkoxyoxamoyl-pyrazines AMERICAN HOME PRODUCTS CORPORATION (US) 1977-07-19 US disclosed
US-3966965-A Oxamic acid derivatives for the prevention of immediate type hypersensitivity reactions AMERICAN HOME PRODUCTS CORPORATION (US) 1976-06-29 US disclosed