SCHEMBL11064121

SCHEMBL11064121

Cc1ccc(Cc2csc(N3CCNCC3)n2)cc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AOC3 Q16853 1/20 0.51
ADRB1 P08588 1/20 0.44
HTR3A P46098 2/20 0.43
SOS1 Q07889 1/20 0.42
BAZ2A Q9UIF9 5/20 0.40
DPP4 P27487 1/20 0.40
CXCR4 P61073 1/20 0.39
POLB P06746 1/20 0.38
SIRT5 Q9NXA8 1/20 0.38
HTR2B P41595 2/20 0.38
HTR2C P28335 1/20 0.38
NMT1 P30419 1/20 0.38
HTR1A P08908 2/20 0.37
CYP1A2 P05177 1/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2D6 P10635 1/20 0.37
CYP2C9 P11712 1/20 0.37
HTR1D P28221 1/20 0.37
HTR1B P28222 1/20 0.37
HTR7 P34969 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11064399 0.86 AOC3 (0.51) AOC3HTR3ASOS1HTR2BHTR2C
SCHEMBL11071226 0.86 CETP (0.51) AOC3ADRB1HTR3ASOS1HTR2B
SCHEMBL3015461 0.86 TAAR1 (0.50) AOC3ADRB1HTR3AHTR6AR
SCHEMBL11065972 0.86 AOC3 (0.48) AOC3ADRB1HTR3APOLBHTR2B
SCHEMBL11071879 0.85 ADRB1 (0.46) AOC3ADRB1HTR3APOLBHTR2B
SCHEMBL11071906 0.84 AOC3 (0.49) AOC3HTR2CHTR1AHTR7HTR6
SCHEMBL11063733 0.82 AOC3 (0.47) AOC3HTR3AHTR2CHTR1ACYP1A2
SCHEMBL11119090 0.81 MAPT (0.52) AOC3ADRB1HTR3ASOS1HTR2B
SCHEMBL11070162 0.81 SCN4A (0.52) AOC3HTR3AHTR1AHTR6CETP
SCHEMBL11066808 0.81 AOC3 (0.48) AOC3ADRB1HTR3ANMT1HTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0005091-B1 MONOSUBSTITUTED PIPERAZINES, PROCESSES FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM SCIENCE UNION ET Cie SOCIETE FRANCAISE DE RECHERCHE MEDICALE (FR) 1981-11-25 EP claimed
US-4479952-A 1-(4-benzyl-2-thiazolyl) piperazine; antiinflammatory; immunomodulator SCIENCE UNION ET CIE (FR) 1984-10-30 US disclosed