SCHEMBL11071879

SCHEMBL11071879

Cc1cccc(Cc2csc(N3CCNCC3)n2)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRB1 P08588 1/20 0.46
AOC3 Q16853 1/20 0.45
HTR6 P50406 5/20 0.44
CTSB P07858 1/20 0.44
CTSS P25774 1/20 0.44
CTSK P43235 1/20 0.44
HTR2C P28335 2/20 0.42
HTR2B P41595 1/20 0.42
OPRL1 P41146 1/20 0.41
HTR1A P08908 3/20 0.40
HTR3A P46098 3/20 0.40
LTA4H P09960 1/20 0.40
DNM1L O00429 1/20 0.39
KHK P50053 1/20 0.39
SLC6A2 P23975 1/20 0.39
SLC6A4 P31645 1/20 0.39
SLC6A3 Q01959 1/20 0.39
MEN1 O00255 1/20 0.39
POLB P06746 1/20 0.39
KMT2A Q03164 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11062910 0.85 HTR2C (0.47) ADRB1AOC3HTR6HTR2CHTR2B
SCHEMBL8067225 0.85 ADRB1 (0.50) ADRB1AOC3HTR6HTR2CHTR2B
SCHEMBL11064121 0.85 AOC3 (0.51) ADRB1AOC3HTR6HTR2CHTR2B
SCHEMBL3015461 0.84 TAAR1 (0.50) ADRB1AOC3HTR6HTR3A
SCHEMBL11062806 0.82 HTR2C (0.50) ADRB1AOC3HTR6HTR2CHTR2B
SCHEMBL2009116 0.79 HTR2C (0.48) ADRB1HTR6CTSBCTSSCTSK
SCHEMBL11066808 0.79 AOC3 (0.48) ADRB1AOC3HTR6HTR1AHTR3A
SCHEMBL11071574 0.79 ERBB2 (0.47) AOC3HTR1AHTR3APOLB
SCHEMBL3009926 0.78 MAPT (0.46) MEN1KMT2A
SCHEMBL11071906 0.78 AOC3 (0.49) AOC3HTR6CTSBCTSSCTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0005091-B1 MONOSUBSTITUTED PIPERAZINES, PROCESSES FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM SCIENCE UNION ET Cie SOCIETE FRANCAISE DE RECHERCHE MEDICALE (FR) 1981-11-25 EP claimed
US-4479952-A 1-(4-benzyl-2-thiazolyl) piperazine; antiinflammatory; immunomodulator SCIENCE UNION ET CIE (FR) 1984-10-30 US disclosed