SCHEMBL11064302

SCHEMBL11064302

CCOC(=O)c1ccccc1C(=O)c1ccc(S(C)(=O)=O)n1CCC1C(=O)OC(C)(C)OC1=O

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 5/20 0.39
CDC25B P30305 1/20 0.36
CYP11B2 P19099 1/20 0.34
ALDH1A1 P00352 4/20 0.33
HSD17B10 Q99714 3/20 0.33
KDM4E B2RXH2 3/20 0.33
LMNA P02545 2/20 0.33
METAP2 P50579 1/20 0.33
MAOB P27338 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
MAPT P10636 2/20 0.33
KMT2A Q03164 2/20 0.33
MEN1 O00255 1/20 0.32
USP2 O75604 1/20 0.32
HPGD P15428 1/20 0.32
TNNI3 P19429 1/20 0.32
CASP1 P29466 1/20 0.32
BRCA1 P38398 1/20 0.32
TNNT2 P45379 1/20 0.32
CASP7 P55210 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11061676 0.79 KAT6A (0.32)
SCHEMBL11055038 0.78 BACE1 (0.32)
SCHEMBL11069050 0.74
SCHEMBL9792244 0.69 MDM2 (0.35) ALDH1A1HSD17B10LMNANPSR1MAPT
SCHEMBL11090292 0.68 ALDH1A1 (0.32) ALDH1A1NPSR1
SCHEMBL11064801 0.67 PTGS2 (0.34) ALDH1A1KDM4ELMNANPSR1
SCHEMBL9792202 0.66 SMN1; SMN2 (0.46) TSHRALDH1A1HSD17B10KDM4ELMNA
SCHEMBL9792291 0.65 MEN1 (0.35) ALDH1A1KMT2AMEN1HPGD
SCHEMBL9792193 0.64 HTT (0.41) LMNAMAPTKMT2AHPGD
SCHEMBL31009568 0.64 TSHR (0.88) TSHRCDC25BALDH1A1HSD17B10KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4458081-A ANTIINFLAMMATORY, ANALGESIC, ANTICOAGULANT, MUSCLE RELAXANT SYNTEX (U.S.A.) INC. (US) 1984-07-03 US disclosed
US-4454326-A 5-Aroyl 6-chloro or 6-bromo 1,2-dihydro-3H-pyrrolo[1,2-a]pyrrole-1,1-di-carboxylates SYNTEX (U.S.A.) INC. (US) 1984-06-12 US disclosed
US-4347187-A Process for preparing 5-aroyl 1,2-dihydro-3H-pyrrolo[1,2-a]pyrrole-1-carboxylic acids and novel intermediates therein SYNTEX (U.S.A.) INC. (US) 1982-08-31 US disclosed
US-4347186-A Process for preparing 5-aroyl 1,2-dihydro-3-H pyrrolo[1,2-a]pyrrole-1-carboxylic acids and novel intermediates therein SYNTEX (U.S.A.) INC. (US) 1982-08-31 US disclosed