SCHEMBL11067253

SCHEMBL11067253

Cc1cccc2c(O)c(CS(C)(=O)=O)cnc12

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 1/20 0.39
HTR1A P08908 1/20 0.38
ADRA1D P25100 1/20 0.38
ADRA1A P35348 1/20 0.38
ADRA1B P35368 1/20 0.38
MEN1 O00255 2/20 0.37
KMT2A Q03164 2/20 0.37
NPC1 O15118 1/20 0.37
RAB9A P51151 1/20 0.37
NR1H2 P55055 2/20 0.37
NR1H3 Q13133 2/20 0.37
CA1 P00915 1/20 0.36
CA2 P00918 1/20 0.36
ELANE P08246 1/20 0.36
PPARG P37231 1/20 0.35
PPARD Q03181 1/20 0.35
PPARA Q07869 1/20 0.35
KDM4E B2RXH2 1/20 0.35
ALDH1A1 P00352 1/20 0.35
LMNA P02545 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11064349 0.79 ERN1 (0.44) CA1CA2KDM4EALDH1A1LMNA
SCHEMBL11067317 0.78 HTR1A (0.39) PARP1HTR1AADRA1DADRA1AADRA1B
SCHEMBL18436554 0.76 ALDH1A1 (0.44) PARP1HTR1AADRA1DADRA1AADRA1B
SCHEMBL29934098 0.75 PARP1 (0.40) PARP1HTR1AADRA1DADRA1AADRA1B
SCHEMBL19692927 0.75 PARP1 (0.40) PARP1HTR1AADRA1DADRA1AADRA1B
Hydrochloric Acid SCHEMBL28291851 0.75 COMT (0.41) PARP1HTR1AADRA1DADRA1AADRA1B
SCHEMBL11061991 0.72 CA1 (0.38) PARP1HTR1AADRA1DADRA1AADRA1B
SCHEMBL28472245 0.71 PARP1 (0.41) PARP1HTR1AADRA1DADRA1AADRA1B
SCHEMBL8123989 0.71 POLB (0.51) PARP1MEN1KMT2AKDM4EALDH1A1
SCHEMBL28815874 0.71 KDM4E (0.51) PARP1MEN1KMT2ANPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4447435-A HYPOTENSIVE AGENTS THE BOOTS COMPANY PLC (GB) 1984-05-08 US disclosed
US-4442109-A 3-Methylthiomethyl-and 3-methylsulfinylmethyl-4-quinolinones useful for treating hypertension THE BOOTS COMPANY LIMITED (GB) 1984-04-10 US disclosed