SCHEMBL11067767

SCHEMBL11067767

O=Cc1c[nH]c2cccc(OCC3CO3)c12

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 2/20 0.47
ALDH1A1 P00352 5/20 0.44
GLA P06280 1/20 0.44
SMN1; SMN2 Q16637 2/20 0.40
TP53 P04637 1/20 0.40
CYP3A4 P08684 1/20 0.40
TSHR P16473 1/20 0.40
HIF1A Q16665 1/20 0.40
TDP1 Q9NUW8 1/20 0.38
IMPDH2 P12268 1/20 0.38
HTR2A P28223 2/20 0.35
HTR2C P28335 1/20 0.35
HTR2B P41595 1/20 0.35
TRIM24 O15164 1/20 0.35
TRIM33 Q9UPN9 1/20 0.35
DRD4 P21917 1/20 0.34
LMNA P02545 1/20 0.34
GAA P10253 1/20 0.34
PKM P14618 1/20 0.34
HTR1D P28221 7/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10338142 0.84 CYP2A6 (0.40) CYP2A6ALDH1A1GLASMN1; SMN2TP53
SCHEMBL11633784 0.80 ALDH1A1 (0.48) ALDH1A1GLASMN1; SMN2TP53CYP3A4
SCHEMBL29950589 0.78 CYP2A6 (0.54) CYP2A6ALDH1A1SMN1; SMN2TDP1IMPDH2
SCHEMBL10505249 0.78 ALDH1A1 (0.46) ALDH1A1GLASMN1; SMN2TP53CYP3A4
SCHEMBL11064847 0.78 ALDH1A1 (0.46) ALDH1A1GLASMN1; SMN2TP53CYP3A4
SCHEMBL28937430 0.76 ALDH1A1 (0.60) ALDH1A1GLASMN1; SMN2TP53CYP3A4
SCHEMBL1034135 0.76 ALDH1A1 (0.60) ALDH1A1GLASMN1; SMN2TP53CYP3A4
SCHEMBL4367638 0.76 ALDH1A1 (0.60) ALDH1A1GLASMN1; SMN2TP53CYP3A4
SCHEMBL1419107 0.75 HTR2A (0.55) CYP2A6SMN1; SMN2TDP1IMPDH2HTR2A
SCHEMBL29954497 0.75 HTR2A (0.55) CYP2A6SMN1; SMN2TDP1IMPDH2HTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0045910-B1 INDOLE DERIVATIVES AND PROCESS FOR THEIR PRODUCTION Roche Diagnostics GmbH (DE) 1984-10-10 EP disclosed
US-4468520-A BETA-BLOCKERS BOEHRINGER MANNHEIM GMBH (DE) 1984-08-28 US disclosed
US-4442295-A 3-Cyano indoles as intermediates for cardioselective compounds BOEHRINGER MANNHEIM GMBH (DE) 1984-04-10 US disclosed
EP-0045911-B1 PROPANOL AMINE, DERIVATIVES, PROCESS FOR THEIR PREPARATION AND MEDICINES CONTAINING THESE COMPOUNDS Roche Diagnostics GmbH (DE) 1983-12-14 EP disclosed
EP-0045911-A1 Propanol amine, derivatives, process for their preparation and medicines containing these compounds Roche Diagnostics GmbH (DE) 1982-02-17 EP disclosed
EP-0045910-A1 Indole derivatives and process for their production Roche Diagnostics GmbH (DE) 1982-02-17 EP disclosed