SCHEMBL11070233

SCHEMBL11070233

CCCCNC(=O)C(C)N1CCNCC1

nearest known ligand 0.60

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 3/20 0.60
USP2 O75604 1/20 0.41
GNAI3 P08754 3/20 0.40
GNAO1 P09471 3/20 0.40
GNAI1 P63096 3/20 0.40
EPHX1 P07099 3/20 0.39
HTT P42858 1/20 0.39
ACHE P22303 2/20 0.39
DPP7 Q9UHL4 1/20 0.38
MEN1 O00255 1/20 0.37
CNR1 P21554 1/20 0.37
CNR2 P34972 1/20 0.37
KMT2A Q03164 1/20 0.37
CHRM5 P08912 1/20 0.37
CHRM3 P20309 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
MMP8 P22894 1/20 0.37
LMNA P02545 1/20 0.37
PAX8 Q06710 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11066224 0.95 SIGMAR1 (0.59) SIGMAR1USP2GNAI3GNAO1GNAI1
SCHEMBL11060304 0.94 SIGMAR1 (0.58) SIGMAR1GNAI3GNAO1GNAI1EPHX1
SCHEMBL11066538 0.90 SIGMAR1 (0.63) SIGMAR1USP2GNAI3GNAO1GNAI1
SCHEMBL1554806 0.90 SIGMAR1 (0.57) SIGMAR1USP2GNAI3GNAO1GNAI1
SCHEMBL6678936 0.83 SIGMAR1 (0.58) SIGMAR1GNAI3GNAO1GNAI1HTT
SCHEMBL8508376 0.81 SIGMAR1 (0.54) SIGMAR1GNAI3GNAO1GNAI1EPHX1
SCHEMBL8508634 0.80 SIGMAR1 (0.59) SIGMAR1CHRM5CHRM3
SCHEMBL11060305 0.79 SIGMAR1 (0.57) SIGMAR1EPHX1MEN1KMT2ACHRM5
SCHEMBL29957416 0.78 SIGMAR1 (0.44) SIGMAR1USP2GNAI3GNAO1GNAI1
SCHEMBL7748187 0.78 SIGMAR1 (0.56) SIGMAR1MEN1KMT2ACHRM5CHRM3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4478838-A VASODILATOR AGENTS HOKURIKU PHARMACEUTICAL CO., LTD. (JP) 1984-10-23 US disclosed
EP-0083712-A1 1-(3,4,5-Trimethoxycinnamoyl)-4-aminocarbonylethyl-substituted piperazine derivatives and a process for the preparation thereof Hokuriku Pharmaceutical Co.,Ltd (JP) 1983-07-20 EP disclosed