SCHEMBL11066538

SCHEMBL11066538

CCCNC(=O)C(C)N1CCNCC1

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 4/20 0.63
CHRM5 P08912 1/20 0.39
CHRM3 P20309 1/20 0.39
OPRD1 P41143 4/20 0.37
GNAI3 P08754 1/20 0.36
GNAO1 P09471 1/20 0.36
GNAI1 P63096 1/20 0.36
CHRNB2 P17787 1/20 0.35
CHRNB4 P30926 1/20 0.35
CHRNA3 P32297 1/20 0.35
CHRNA7 P36544 1/20 0.35
CHRNA4 P43681 1/20 0.35
OPRM1 P35372 3/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
HSD17B10 Q99714 1/20 0.34
USP2 O75604 2/20 0.34
KDM4E B2RXH2 2/20 0.34
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
TSHR P16473 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11070233 0.90 SIGMAR1 (0.60) SIGMAR1CHRM5CHRM3GNAI3GNAO1
SCHEMBL11066224 0.89 SIGMAR1 (0.59) SIGMAR1GNAI3GNAO1GNAI1USP2
SCHEMBL11060304 0.88 SIGMAR1 (0.58) SIGMAR1GNAI3GNAO1GNAI1
SCHEMBL6678936 0.86 SIGMAR1 (0.58) SIGMAR1CHRM5CHRM3OPRD1GNAI3
SCHEMBL1554806 0.84 SIGMAR1 (0.57) SIGMAR1OPRD1GNAI3GNAO1GNAI1
SCHEMBL4559647 0.83 SIGMAR1 (0.46) SIGMAR1CHRM5CHRM3OPRD1GNAI3
SCHEMBL8508634 0.83 SIGMAR1 (0.59) SIGMAR1CHRM5CHRM3OPRD1SMN1; SMN2
SCHEMBL11060305 0.81 SIGMAR1 (0.57) SIGMAR1CHRM5CHRM3OPRD1OPRM1
SCHEMBL1907641 0.81 SIGMAR1 (0.44) SIGMAR1CHRM5CHRM3OPRD1GNAI3
SCHEMBL7748187 0.80 SIGMAR1 (0.56) SIGMAR1CHRM5CHRM3OPRD1OPRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4478838-A VASODILATOR AGENTS HOKURIKU PHARMACEUTICAL CO., LTD. (JP) 1984-10-23 US disclosed
EP-0083712-A1 1-(3,4,5-Trimethoxycinnamoyl)-4-aminocarbonylethyl-substituted piperazine derivatives and a process for the preparation thereof Hokuriku Pharmaceutical Co.,Ltd (JP) 1983-07-20 EP disclosed