SCHEMBL11070834

SCHEMBL11070834

COc1ccccc1OC(CCc1ccc(C)cc1)Cn1ccnc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP11B1 P15538 2/20 0.45
CYP11B2 P19099 2/20 0.45
CYP19A1 P11511 2/20 0.45
TBXAS1 P24557 1/20 0.44
FNTA P49354 1/20 0.43
FNTB P49356 1/20 0.43
PGGT1B P53609 1/20 0.43
ALDH1A1 P00352 3/20 0.42
CYP3A4 P08684 3/20 0.42
TDP1 Q9NUW8 3/20 0.42
TP53 P04637 2/20 0.42
CYP1A2 P05177 2/20 0.42
CYP2C9 P11712 2/20 0.42
TSHR P16473 2/20 0.42
MAPT P10636 2/20 0.42
LMNA P02545 1/20 0.42
CYP2D6 P10635 1/20 0.42
ALOX15 P16050 1/20 0.42
CYP2C19 P33261 1/20 0.42
HIF1A Q16665 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11077224 0.91 TBXAS1 (0.55) CYP19A1TBXAS1ALDH1A1CYP3A4TDP1
SCHEMBL11070016 0.90 ALDH1A1 (0.53) CYP11B1CYP11B2CYP19A1TBXAS1FNTA
SCHEMBL11068769 0.88 IDO1 (0.43) CYP11B1CYP11B2CYP19A1TBXAS1FNTA
SCHEMBL11066434 0.86 IDO1 (0.50) CYP11B1CYP11B2CYP19A1TBXAS1ALDH1A1
SCHEMBL11079547 0.86 TBXAS1 (0.45) CYP11B1CYP11B2CYP19A1TBXAS1FNTA
SCHEMBL11087691 0.86 IDO1 (0.50) CYP11B1CYP11B2CYP19A1TBXAS1ALDH1A1
SCHEMBL11067638 0.85 TBXAS1 (0.53) CYP19A1TBXAS1ALDH1A1CYP3A4TDP1
SCHEMBL11080068 0.84 TBXAS1 (0.57) CYP11B1CYP11B2CYP19A1TBXAS1ALDH1A1
SCHEMBL11076903 0.82 TBXAS1 (0.52) CYP19A1TBXAS1ALDH1A1CYP3A4TDP1
SCHEMBL11077447 0.82 TBXAS1 (0.52) CYP19A1TBXAS1ALDH1A1CYP3A4TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0005980-B1 DERIVATIVES OF SUBSTITUTED N-ALKYL IMIDAZOLES, THEIR PREPARATION AND THESE COMPOUNDS FOR PHARMACEUTICAL USE SYNTEX (U.S.A.) INC. (US) 1984-08-29 EP disclosed
US-4213991-A BACTERICIDES, FUNGICIDES, ANTIPROTOZOA SYNTEX (U.S.A.) INC. (US) 1980-07-22 US disclosed
EP-0005980-A2 Derivatives of substituted N-alkyl imidazoles, their preparation and these compounds for pharmaceutical use SYNTEX (U.S.A.) INC. (US) 1979-12-12 EP disclosed