SCHEMBL11071068

SCHEMBL11071068

NCC(=O)NC1CCN(CCc2c[nH]c3ccccc23)CC1

nearest known ligand 0.74

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRA2A P08913 1/20 0.74
ADRA2B P18089 1/20 0.74
ADRA2C P18825 1/20 0.74
ADRA1D P25100 1/20 0.74
ADRA1A P35348 1/20 0.74
ADRA1B P35368 1/20 0.74
BCHE P06276 2/20 0.65
ACHE P22303 2/20 0.65
HPGD P15428 1/20 0.63
HTT P42858 1/20 0.63
RECQL P46063 1/20 0.63
SIGMAR1 Q99720 2/20 0.62
HDAC8 Q9BY41 1/20 0.59
HDAC6 Q9UBN7 1/20 0.59
HTR2A P28223 1/20 0.57
SOS1 Q07889 5/20 0.57
KRAS P01116 1/20 0.57
HTR1A P08908 1/20 0.51
NPC1 O15118 1/20 0.51
RAB9A P51151 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11068159 0.89 ADRA2A (0.77) ADRA2AADRA2BADRA2CADRA1DADRA1A
SCHEMBL20812407 0.89 SIGMAR1 (0.71) ADRA2AADRA2BADRA2CADRA1DADRA1A
SCHEMBL11462973 0.89 ADRA2A (0.77) ADRA2AADRA2BADRA2CADRA1DADRA1A
SCHEMBL14564212 0.87 SIGMAR1 (0.62) ADRA2AADRA2BADRA2CADRA1DADRA1A
SCHEMBL10854033 0.87 ADRA2A (0.77) ADRA2AADRA2BADRA2CADRA1DADRA1A
Hydrochloric Acid SCHEMBL5445668 0.86 SIGMAR1 (0.61) ADRA2AADRA2BADRA2CADRA1DADRA1A
Hydrochloric Acid SCHEMBL5445673 0.86 SIGMAR1 (0.61) ADRA2AADRA2BADRA2CADRA1DADRA1A
SCHEMBL11548936 0.85 ADRA2A (0.74) ADRA2AADRA2BADRA2CADRA1DADRA1A
SCHEMBL11547157 0.85 ADRA2A (0.74) ADRA2AADRA2BADRA2CADRA1DADRA1A
SCHEMBL10783732 0.85 ADRA2A (0.80) ADRA2AADRA2BADRA2CADRA1DADRA1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4443461-A N-[2-[[1-[1H-Indolylalkyl- or oxoalkyl]-4-piperidinyl]-amino]-2-oxoethyl]-arylcarboxamide derivatives JOHN WYETH & BROTHER LIMITED (GB) 1984-04-17 US disclosed