SCHEMBL11071083

SCHEMBL11071083

CC(C)(C)Oc1ccc(CCC(Cn2ccnc2)Oc2ccc(Cl)cc2Cl)cc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 6/20 0.53
CYP2C9 P11712 6/20 0.53
IDO1 P14902 8/20 0.46
CYP1A2 P05177 5/20 0.44
CYP2D6 P10635 5/20 0.44
CYP2C19 P33261 5/20 0.44
NR1I2 O75469 3/20 0.44
NR3C1 P04150 3/20 0.44
ADORA3 P0DMS8 3/20 0.44
ADRA2B P18089 3/20 0.44
CHRM3 P20309 3/20 0.44
OPRK1 P41145 3/20 0.44
SLC6A3 Q01959 3/20 0.44
PDE4D Q08499 3/20 0.44
KCNH2 Q12809 3/20 0.44
ALOX15 P16050 3/20 0.44
TDP1 Q9NUW8 3/20 0.44
ADRA2C P18825 3/20 0.44
FYN P06241 2/20 0.44
CHRM4 P08173 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11071440 0.93 IDO1 (0.44) CYP3A4CYP2C9IDO1CYP1A2CYP2D6
SCHEMBL11079557 0.89 IDO1 (0.58) CYP3A4CYP2C9IDO1CYP1A2CYP2D6
SCHEMBL11632605 0.89 CYP3A4 (0.61) CYP3A4CYP2C9IDO1CYP1A2CYP2D6
SCHEMBL11078515 0.89 ALDH1A1 (0.45) CYP3A4CYP2C9CYP1A2CYP2D6CYP2C19
SCHEMBL11070048 0.85 IDO1 (0.51) CYP3A4CYP2C9IDO1CYP1A2CYP2D6
SCHEMBL11076362 0.84 TDP1 (0.45) CYP3A4CYP2C9CYP1A2TDP1TBXAS1
SCHEMBL11081326 0.83 ALDH1A1 (0.48) CYP3A4CYP2C9CYP1A2CYP2D6CYP2C19
SCHEMBL11079547 0.82 TBXAS1 (0.45) CYP3A4CYP2C9CYP1A2CYP2D6CYP2C19
SCHEMBL11070372 0.82 IDO1 (0.56) CYP3A4CYP2C9IDO1CYP1A2CYP2D6
SCHEMBL11070658 0.82 MEN1 (0.41) CYP3A4CYP2C9CYP1A2TDP1TBXAS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0005980-B1 DERIVATIVES OF SUBSTITUTED N-ALKYL IMIDAZOLES, THEIR PREPARATION AND THESE COMPOUNDS FOR PHARMACEUTICAL USE SYNTEX (U.S.A.) INC. (US) 1984-08-29 EP disclosed
US-4213991-A BACTERICIDES, FUNGICIDES, ANTIPROTOZOA SYNTEX (U.S.A.) INC. (US) 1980-07-22 US disclosed