SCHEMBL11072135

SCHEMBL11072135

CC(C)c1nc2c([nH]1)N(CCOc1ccccc1)C1=NCCN1C2=O

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 3/20 0.43
KMT2A Q03164 3/20 0.43
PLA2G7 Q13093 2/20 0.38
ALDH1A1 P00352 4/20 0.38
MAPT P10636 3/20 0.38
APOBEC3A P31941 1/20 0.38
RECQL P46063 1/20 0.38
APOBEC3G Q9HC16 1/20 0.38
GAA P10253 1/20 0.38
TP53 P04637 1/20 0.36
RAB9A P51151 2/20 0.36
NPC1 O15118 1/20 0.36
MAPK1 P28482 2/20 0.35
LMNA P02545 2/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
TSHR P16473 1/20 0.35
HPGD P15428 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
HTR2C P28335 1/20 0.34
CYP3A4 P08684 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10800850 0.87 KMT2A (0.45) MEN1KMT2APLA2G7ALDH1A1MAPT
SCHEMBL11125673 0.80 MEN1 (0.45) MEN1KMT2APLA2G7ALDH1A1MAPT
SCHEMBL10800856 0.75 KMT2A (0.45) MEN1KMT2APLA2G7ALDH1A1MAPT
SCHEMBL10800874 0.70 MEN1 (0.45) MEN1KMT2APLA2G7ALDH1A1MAPT
SCHEMBL11067241 0.70 TSHR (0.42) MEN1KMT2AALDH1A1GAATP53
SCHEMBL11063263 0.66 CYP3A4 (0.32) LMNATSHRCYP3A4SMN1; SMN2HIF1A
SCHEMBL11067126 0.63 MEN1 (0.46) MEN1KMT2AALDH1A1LMNATSHR
SCHEMBL10798396 0.62 TSHR (0.55) MEN1KMT2AGAATP53TSHR
SCHEMBL11070883 0.61 MEN1 (0.44) MEN1KMT2AALDH1A1LMNATSHR
SCHEMBL11842041 0.59 TSHR (0.60) MEN1KMT2AALDH1A1GAALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4489078-A Diazaheterocyclopurines used as anti-broncho spasmatics and vasodilators MEAD JOHNSON & COMPANY (US) 1984-12-18 US claimed
US-4366156-A Antiallergic methods using diazaheterocyclopurines MEAD JOHNSON & COMPANY (US) 1982-12-28 US claimed
US-4298734-A PHOSPHODIESTERASE INHIBITORS, BRONCHODILATORS, PERIPHERAL VASODILATORS MEAD JOHNSON & COMPANY (US) 1981-11-03 US claimed