SCHEMBL11063263

SCHEMBL11063263

Cc1nc2c([nH]1)N(CC(C)C)C1=NCCN1C2=O

nearest known ligand 0.32

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
HIF1A Q16665 1/20 0.32
PDE1A P54750 2/20 0.32
PDE1B Q01064 2/20 0.32
PDE1C Q14123 2/20 0.32
PDE2A O00408 1/20 0.32
TSHR P16473 3/20 0.31
PDE5A O76074 1/20 0.31
LMNA P02545 1/20 0.30
CYP2D6 P10635 1/20 0.30
DRD2 P14416 1/20 0.30
DRD3 P35462 1/20 0.30
KCNH2 Q12809 1/20 0.30
CLPP Q16740 1/20 0.30
GPR132 Q9UNW8 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11273417 0.86 CYP3A4 (0.32) CYP3A4SMN1; SMN2HIF1ATSHR
SCHEMBL11067126 0.80 MEN1 (0.46) TSHRLMNACYP2D6
SCHEMBL10800851 0.78 P2RX7 (0.35) PDE1APDE1BPDE1CPDE2A
SCHEMBL10798396 0.78 TSHR (0.55) CYP3A4SMN1; SMN2HIF1ATSHRCYP2D6
SCHEMBL10800850 0.74 KMT2A (0.45) CYP3A4SMN1; SMN2HIF1ATSHRLMNA
SCHEMBL11070880 0.70 MEN1 (0.44) TSHRLMNACYP2D6
SCHEMBL10800858 0.68 TSHR (0.33) CYP3A4SMN1; SMN2HIF1ATSHRLMNA
SCHEMBL11089172 0.68 ADORA2A (0.36) CYP3A4SMN1; SMN2HIF1APDE1APDE1B
SCHEMBL11072135 0.66 MEN1 (0.43) CYP3A4SMN1; SMN2HIF1ATSHRLMNA
SCHEMBL10798493 0.65 TSHR (0.54) CYP3A4SMN1; SMN2HIF1ATSHRLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4489078-A Diazaheterocyclopurines used as anti-broncho spasmatics and vasodilators MEAD JOHNSON & COMPANY (US) 1984-12-18 US claimed
US-4366156-A Antiallergic methods using diazaheterocyclopurines MEAD JOHNSON & COMPANY (US) 1982-12-28 US claimed
US-4298734-A PHOSPHODIESTERASE INHIBITORS, BRONCHODILATORS, PERIPHERAL VASODILATORS MEAD JOHNSON & COMPANY (US) 1981-11-03 US claimed