SCHEMBL10798396

SCHEMBL10798396

Cc1nc2c([nH]1)N(Cc1ccc(Cl)cc1)C1=NCCN1C2=O

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 5/20 0.55
HTT P42858 2/20 0.41
CLPP Q16740 4/20 0.39
GAA P10253 1/20 0.38
GFER P55789 1/20 0.38
CYP3A4 P08684 2/20 0.38
TP53 P04637 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
HIF1A Q16665 1/20 0.38
KMT2A Q03164 2/20 0.37
GPR132 Q9UNW8 2/20 0.35
CYP2D6 P10635 1/20 0.35
DRD2 P14416 1/20 0.35
DRD3 P35462 1/20 0.35
KCNH2 Q12809 1/20 0.35
TYMS P04818 1/20 0.35
P2RX7 Q99572 1/20 0.34
POLB P06746 1/20 0.34
PRKAG1 P54619 1/20 0.34
PRKAA1 Q13131 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10798493 0.88 TSHR (0.54) TSHRHTTCLPPGAAGFER
SCHEMBL10795244 0.87 TSHR (0.55) TSHRHTTCLPPGAAGFER
SCHEMBL10798400 0.84 TSHR (0.55) TSHRHTTCLPPGAAGFER
SCHEMBL10800871 0.84 TSHR (0.52) TSHRHTTCLPPGAAGFER
SCHEMBL10800868 0.81 P2RX7 (0.42) TSHRP2RX7
SCHEMBL10795837 0.81 PDE5A (0.35) TSHRHTTKMT2ATYMSP2RX7
SCHEMBL10795586 0.80 TSHR (0.57) TSHRHTTCLPPGAAGFER
Hydrochloric Acid SCHEMBL11069993 0.79 TSHR (0.56) TSHRHTTCLPPGAAGFER
SCHEMBL11063263 0.78 CYP3A4 (0.32) TSHRCLPPCYP3A4SMN1; SMN2HIF1A
SCHEMBL11163356 0.77 TSHR (0.57) TSHRHTTCLPPGAAGFER

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4489078-A Diazaheterocyclopurines used as anti-broncho spasmatics and vasodilators MEAD JOHNSON & COMPANY (US) 1984-12-18 US claimed
US-4366156-A Antiallergic methods using diazaheterocyclopurines MEAD JOHNSON & COMPANY (US) 1982-12-28 US claimed
US-4642345-A BRONCHODILATOR AGENTS MEAD JOHNSON & COMPANY (US) 1987-02-10 US disclosed
US-4489078-A Diazaheterocyclopurines used as anti-broncho spasmatics and vasodilators MEAD JOHNSON & COMPANY (US) 1984-12-18 US disclosed
US-4366156-A Antiallergic methods using diazaheterocyclopurines MEAD JOHNSON & COMPANY (US) 1982-12-28 US disclosed