SCHEMBL11072802

SCHEMBL11072802

CCOC(=O)C(=O)c1cc(CBr)c(C(=O)OCC)[nH]1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.41
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41
LMNA P02545 2/20 0.40
HPGD P15428 4/20 0.39
ALOX15 P16050 1/20 0.38
NPC1 O15118 3/20 0.38
GAA P10253 3/20 0.38
POLB P06746 1/20 0.38
ALDH1A1 P00352 8/20 0.37
MAPT P10636 5/20 0.37
KDM4E B2RXH2 5/20 0.37
RAB9A P51151 3/20 0.37
SMN1; SMN2 Q16637 2/20 0.37
TP53 P04637 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
MAPK1 P28482 1/20 0.37
HSD17B10 Q99714 1/20 0.37
CYP4F2 P78329 1/20 0.37
CYP4A11 Q02928 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11205491 0.71 CYP1A2 (0.47) CYP1A2CYP2C9CYP2C19LMNAHPGD
SCHEMBL11649989 0.68 ALDH1A1 (0.51) CYP1A2CYP2C9CYP2C19LMNAHPGD
SCHEMBL11191069 0.68 CYP1A2 (0.55) CYP1A2CYP2C9CYP2C19LMNAHPGD
SCHEMBL11064802 0.68 CA12 (0.41) LMNAHPGDGAAALDH1A1MAPT
SCHEMBL5443501 0.67 CYP1A2 (0.49) CYP1A2CYP2C9CYP2C19LMNAHPGD
SCHEMBL27034946 0.67 HRH3 (0.50) CYP1A2CYP2C9CYP2C19LMNAHPGD
SCHEMBL2813572 0.66 CYP4F2 (0.53) LMNAHPGDNPC1GAAPOLB
SCHEMBL3023118 0.66 ALDH1A1 (0.54) CYP1A2CYP2C9CYP2C19LMNAHPGD
SCHEMBL10003063 0.66 ALDH1A1 (0.48) CYP1A2CYP2C9CYP2C19LMNAHPGD
SCHEMBL3152177 0.66 ALDH1A1 (0.47) CYP1A2CYP2C9CYP2C19LMNAHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4440779-A Tricyclic derivatives of substituted pyrrole acids as analgesic and anti-inflammatory agents MERCK & CO., INC. (US) 1984-04-03 US disclosed
EP-0068460-A1 Tricyclic derivatives of substituted pyrrole acids as analgesic and anti-inflammatory agents MERCK & CO. INC. (US) 1983-01-05 EP disclosed