SCHEMBL11064802

SCHEMBL11064802

CCOC(=O)C(=O)c1cc(CBr)c(C(=O)OCC)n1C

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 5/20 0.41
CA1 P00915 5/20 0.41
CA2 P00918 5/20 0.41
CA7 P43166 5/20 0.41
CA9 Q16790 5/20 0.41
CA14 Q9ULX7 5/20 0.41
KMT2A Q03164 2/20 0.40
ESR1 P03372 1/20 0.37
ESR2 Q92731 1/20 0.37
KDM4E B2RXH2 2/20 0.37
LMNA P02545 1/20 0.37
HTT P42858 1/20 0.36
ATM Q13315 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
NR1H2 P55055 1/20 0.36
NR1H3 Q13133 1/20 0.36
CYP4F2 P78329 1/20 0.36
CYP4A11 Q02928 1/20 0.36
GAA P10253 3/20 0.35
MAPT P10636 3/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11064170 0.82 HTT (0.46) CA12CA1CA2CA7CA9
SCHEMBL15100671 0.80 ALDH1A1 (0.45) KMT2AKDM4EGAAMAPTALDH1A1
SCHEMBL11063339 0.75 RXRA (0.43) KMT2ALMNAHTTL3MBTL1
SCHEMBL11059944 0.74 ALOX5 (0.54) KMT2ALMNAHTTGAAMAPT
SCHEMBL21408332 0.74 NPSR1 (0.45) CA12CA1CA2CA7CA9
SCHEMBL21428060 0.69 ALDH1A1 (0.43) CA12CA1CA2CA7CA9
SCHEMBL11195139 0.69 KMT2A (0.49) CA12CA1CA2CA7CA9
SCHEMBL21266562 0.68 RAB9A (0.46) CA12CA1CA2CA7CA9
SCHEMBL7702111 0.68 KMT2A (0.44) CA12CA1CA2CA7CA9
SCHEMBL11072802 0.68 CYP1A2 (0.41) KMT2AKDM4ELMNAL3MBTL1CYP4F2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4440779-A Tricyclic derivatives of substituted pyrrole acids as analgesic and anti-inflammatory agents MERCK & CO., INC. (US) 1984-04-03 US disclosed