SCHEMBL11075217

SCHEMBL11075217

COc1ccc(CCC(Cn2ccnc2)Oc2ccc(OC)cc2)cc1

nearest known ligand 0.61

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
TBXAS1 P24557 12/20 0.61
ALDH1A1 P00352 2/20 0.58
CYP3A4 P08684 2/20 0.58
MAPT P10636 2/20 0.58
TDP1 Q9NUW8 2/20 0.58
MEN1 O00255 1/20 0.58
TP53 P04637 1/20 0.58
CYP1A2 P05177 1/20 0.58
TSHR P16473 1/20 0.58
MAPK1 P28482 1/20 0.58
KMT2A Q03164 1/20 0.58
HSD17B10 Q99714 1/20 0.58
CYP2C9 P11712 1/20 0.58
SMN1; SMN2 Q16637 1/20 0.58
TRPM8 Q7Z2W7 1/20 0.58
ORAI1 Q96D31 1/20 0.57
CYP19A1 P11511 2/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11080068 0.95 TBXAS1 (0.57) TBXAS1ALDH1A1CYP3A4MAPTTDP1
SCHEMBL11070590 0.94 TBXAS1 (0.56) TBXAS1ALDH1A1CYP3A4MAPTTDP1
SCHEMBL11068886 0.94 TBXAS1 (0.56) TBXAS1ALDH1A1CYP3A4MAPTTDP1
SCHEMBL10925643 0.94 TBXAS1 (0.56) TBXAS1ALDH1A1CYP3A4MAPTTDP1
SCHEMBL10930745 0.92 TBXAS1 (0.54) TBXAS1ALDH1A1CYP3A4MAPTTDP1
SCHEMBL10927229 0.89 TBXAS1 (0.51) TBXAS1ALDH1A1CYP3A4MAPTTDP1
SCHEMBL10928025 0.89 TBXAS1 (0.51) TBXAS1ALDH1A1CYP3A4MAPTTDP1
SCHEMBL10925479 0.89 TBXAS1 (0.51) TBXAS1ALDH1A1CYP3A4MAPTTDP1
SCHEMBL11077224 0.88 TBXAS1 (0.55) TBXAS1ALDH1A1CYP3A4MAPTTDP1
Hydrochloric Acid SCHEMBL10927733 0.87 RAB9A (0.55) TBXAS1ALDH1A1CYP3A4MAPTTDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0005980-B1 DERIVATIVES OF SUBSTITUTED N-ALKYL IMIDAZOLES, THEIR PREPARATION AND THESE COMPOUNDS FOR PHARMACEUTICAL USE SYNTEX (U.S.A.) INC. (US) 1984-08-29 EP disclosed
US-4213991-A BACTERICIDES, FUNGICIDES, ANTIPROTOZOA SYNTEX (U.S.A.) INC. (US) 1980-07-22 US disclosed
EP-0005980-A2 Derivatives of substituted N-alkyl imidazoles, their preparation and these compounds for pharmaceutical use SYNTEX (U.S.A.) INC. (US) 1979-12-12 EP disclosed