SCHEMBL11075409

SCHEMBL11075409

C=CCN1CCCC1CNC(=O)c1cc(NS(C)(=O)=O)c(C)cc1OC

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 12/20 0.64
DRD3 P35462 10/20 0.64
DRD4 P21917 7/20 0.64
ADRA2B P18089 3/20 0.61
ADRA2C P18825 3/20 0.61
KCNH2 Q12809 3/20 0.61
HRH3 Q9Y5N1 3/20 0.61
ADRA2A P08913 3/20 0.61
CA2 P00918 3/20 0.61
CA9 Q16790 3/20 0.61
HTR2A P28223 2/20 0.61
SLC6A4 P31645 2/20 0.61
CA12 O43570 2/20 0.61
CA1 P00915 2/20 0.61
DRD1 P21728 2/20 0.61
CA6 P23280 2/20 0.61
CA5A P35218 2/20 0.61
CA7 P43166 2/20 0.61
CA5B Q9Y2D0 2/20 0.61
HTR1A P08908 1/20 0.61

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11090475 0.90 DRD2 (0.63) DRD2DRD3DRD4ADRA2BADRA2C
SCHEMBL11079730 0.90 DRD2 (0.65) DRD2DRD3DRD4ADRA2BADRA2C
SCHEMBL11083763 0.84 SIGMAR1 (0.57) DRD2DRD3DRD4ADRA2BADRA2C
SCHEMBL11084539 0.83 DRD2 (0.68) DRD2DRD3DRD4ADRA2BADRA2C
SCHEMBL11085879 0.83 DRD2 (0.65) DRD2DRD3DRD4ADRA2BADRA2C
SCHEMBL9835471 0.83 DRD2 (0.69) DRD2DRD3DRD4ADRA2BADRA2C
SCHEMBL11090817 0.82 DRD2 (0.66) DRD2DRD3DRD4ADRA2BADRA2C
SCHEMBL11086951 0.82 DRD2 (0.66) DRD2DRD3DRD4ADRA2BADRA2C
SCHEMBL11238878 0.81 DRD2 (0.66) DRD2DRD3DRD4ADRA2BADRA2C
SCHEMBL11090818 0.80 TSHR (0.65) DRD2DRD3DRD4ADRA2BADRA2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4350635-A ANTIEMETICS, NEUROLEPTIC AGENTS SHIONOGI & CO., LTD. (JP) 1982-09-21 US claimed
US-4431663-A ANTIULCER AND NEUROLEPTIC AGENTS; ANTIEMETICS SHIONOGI & CO., LTD. (JP) 1984-02-14 US disclosed
US-4351770-A Preparation of N(2-pyrrolidinylmethyl)2-methoxy-5-benzenesulfonamidobenzamides SHIONOGI & CO., LTD. (JP) 1982-09-28 US disclosed
US-4350635-A ANTIEMETICS, NEUROLEPTIC AGENTS SHIONOGI & CO., LTD. (JP) 1982-09-21 US disclosed
US-4330472-A Meta-sulfonamido-benzamide derivatives SHIONOGI & CO., LTD. (JP) 1982-05-18 US disclosed
US-4328155-A ANTIEMETIC OR PSYCHOTROPIC AGENT SHIONOGI & CO., LTD. (JP) 1982-05-04 US disclosed
US-4328344-A ANTIEMETIC SHIONOGI & CO., LTD. (JP) 1982-05-04 US disclosed