SCHEMBL11076092

SCHEMBL11076092

C=CCN(CCC)C1CCC(c2ccc(CCCC)cc2C)(N(C)C)CC1

nearest known ligand 0.38

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HTR1D P28221 1/20 0.38
SKP2 Q13309 1/20 0.35
HTR1B P28222 1/20 0.34
DRD3 P35462 13/20 0.34
DRD2 P14416 10/20 0.34
CYP1A2 P05177 1/20 0.32
CYP3A4 P08684 1/20 0.32
CYP2D6 P10635 1/20 0.32
CYP2C9 P11712 1/20 0.32
CYP2C19 P33261 1/20 0.32
CYP4Z1 Q86W10 1/20 0.32
CYP4F11 Q9HBI6 1/20 0.32
CYP4F12 Q9HCS2 1/20 0.32
HTR1A P08908 1/20 0.31
SPHK1 Q9NYA1 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11071470 0.81 SKP2 (0.40) SKP2DRD3DRD2CYP1A2CYP3A4
SCHEMBL11076941 0.81 HTR1D (0.40) HTR1DHTR1BDRD3DRD2HTR1A
SCHEMBL11069677 0.81 HTR1D (0.37) HTR1DHTR1BDRD3DRD2CYP1A2
SCHEMBL11074078 0.80 GRIN2B (0.40) SKP2DRD3DRD2
SCHEMBL11070718 0.79 SKP2 (0.35) SKP2CYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL11071467 0.74 SKP2 (0.38) SKP2CYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL11074417 0.73 SKP2 (0.43) SKP2CYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL11076865 0.72 HTR1D (0.36) HTR1DHTR1BDRD3DRD2CYP1A2
SCHEMBL11076134 0.72 HTR1D (0.38) HTR1DHTR1BHTR1A
SCHEMBL11066576 0.72 OPRL1 (0.36) SKP2CYP1A2CYP3A4CYP2D6CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4447454-A Analgetic compounds, compositions and process of treatment THE UPJOHN COMPANY (US) 1984-05-08 US disclosed
US-4113866-A ANALGETIC COMPOUNDS, COMPOSITIONS AND PROCESS OF TREATMENT THE UPJOHN COMPANY (US) 1978-09-12 US disclosed