SCHEMBL11078611

SCHEMBL11078611

C[S+]([O-])c1cccc([S+](C)[O-])c1C(CC(N)=O)CC(N)=O

nearest known ligand 0.35

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
CYP2C19 P33261 2/20 0.31
ITGB2 P05107 1/20 0.31
ICAM1 P05362 1/20 0.31
ITGAL P20701 1/20 0.31
CYP1A2 P05177 1/20 0.31
CYP2D6 P10635 1/20 0.31
PKM P14618 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
NPSR1 Q6W5P4 1/20 0.31
KDM4E B2RXH2 1/20 0.30
MAPT P10636 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11076201 0.77
SCHEMBL11074850 0.75 MMP2 (0.32)
SCHEMBL11078116 0.71 ALDH1A1 (0.42) ALDH1A1L3MBTL1CYP2C19CYP1A2CYP2D6
SCHEMBL11074706 0.69 ITGB2 (0.43) ALDH1A1CYP2C19ITGB2ICAM1ITGAL
SCHEMBL11075085 0.69 ALDH1A1 (0.36) ALDH1A1L3MBTL1CYP2C19ITGB2ICAM1
SCHEMBL11071260 0.69 ITGB2 (0.38) ALDH1A1L3MBTL1CYP2C19ITGB2ICAM1
SCHEMBL11079548 0.69 ITGB2 (0.49) ALDH1A1L3MBTL1ITGB2ICAM1ITGAL
SCHEMBL11076609 0.69 ESR1 (0.31)
SCHEMBL11084188 0.69
SCHEMBL11076456 0.68 CYP1A2 (0.37) ALDH1A1L3MBTL1CYP2C19ITGB2ICAM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0024776-B1 4-PHENYL AND 5-PHENYL-1,4,5,6-TETRAHYDROPYRIMIDINE DERIVATIVES, PHARMACEUTICAL COMPOSITIONS CONTAINING SAID DERIVATIVES, AND PROCESS FOR PREPARING SAID DERIVATIVES SYNTEX (U.S.A.) INC. (US) 1984-12-27 EP disclosed
US-4322421-A 4-Phenyl-and 5-phenyl-1,4,5,6-tetrahydro-pyrimidine derivatives SYNTEX (U.S.A.) INC. (US) 1982-03-30 US disclosed
US-4261995-A DISORDERS OF CENTRAL NERVOUS SYSTEM AND CARDIOVASCULAR SYSTEM; HYPOTENSIVE SYNTEX (U.S.A.) INC. (US) 1981-04-14 US disclosed
EP-0024776-A1 4-Phenyl and 5-phenyl-1,4,5,6-tetrahydropyrimidine derivatives, pharmaceutical compositions containing said derivatives, and process for preparing said derivatives SYNTEX (U.S.A.) INC. (US) 1981-03-11 EP disclosed