SCHEMBL11079176

SCHEMBL11079176

CC(=O)NC1CN(S(=O)(=O)O)C1=O.c1cc2cc-2c1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 4/20 0.37
CA2 P00918 4/20 0.37
CA12 O43570 3/20 0.37
CA7 P43166 3/20 0.37
CA14 Q9ULX7 3/20 0.37
CA9 Q16790 2/20 0.37
IRAK4 Q9NWZ3 2/20 0.35
KDM4E B2RXH2 2/20 0.34
MAPT P10636 2/20 0.34
ALDH1A1 P00352 2/20 0.34
THRB P10828 1/20 0.34
HSD17B10 Q99714 1/20 0.34
LMNA P02545 1/20 0.34
POLB P06746 1/20 0.34
GRIA2 P42262 3/20 0.34
KCNH2 Q12809 2/20 0.34
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
IRAK1 P51617 1/20 0.32
AKR1C3 P42330 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Pyridine SCHEMBL10680880 0.92 ALDH1A1 (0.34) CA1CA2CA12CA7CA14
SCHEMBL10678594 0.87 NSD2 (0.34) CA1CA2CA12CA7CA14
SCHEMBL10678605 0.87 NSD2 (0.34) CA1CA2CA12CA7CA14
SCHEMBL10545523 0.87 CA1 (0.38) CA1CA2CA12CA7CA14
SCHEMBL10653301 0.80 IRAK4 (0.37) CA1CA2CA12CA7CA14
SCHEMBL10649367 0.76 KDM4E (0.36) CA1CA2CA12CA7CA14
SCHEMBL10860123 0.75 ACE (0.42) KDM4EALDH1A1
SCHEMBL8895550 0.75 MEN1 (0.34) CA1CA2CA12CA7CA14
SCHEMBL11293989 0.74 IRAK4 (0.36) IRAK4KDM4EMAPTALDH1A1THRB
SCHEMBL10674812 0.73 PTGS1 (0.43) CA1CA2CA12CA7CA14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0021678-B1 1-SULPHO-2-OXOAZETIDINE DERIVATIVES, THEIR PRODUCTION AND PHARMACEUTICAL COMPOSITIONS THEREOF Takeda Chemical Industries, Ltd. (JP) 1984-11-07 EP claimed
JP-55164672-A None JP disclosed
JP-S55164672-A AZETIDINE DERIVATIVE AND ITS PREPARATION TAKEDA CHEM IND LTD 1980-12-22 JP disclosed