SCHEMBL10653301

SCHEMBL10653301

CC(=O)NC1CN(O)C1=O.c1cc2cc-2c1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IRAK4 Q9NWZ3 2/20 0.37
KDM4E B2RXH2 3/20 0.37
ALDH1A1 P00352 3/20 0.37
MAPT P10636 2/20 0.37
THRB P10828 1/20 0.37
HSD17B10 Q99714 1/20 0.37
LMNA P02545 1/20 0.36
POLB P06746 1/20 0.36
CA12 O43570 1/20 0.35
CA1 P00915 1/20 0.35
CA2 P00918 1/20 0.35
CA7 P43166 1/20 0.35
CA9 Q16790 1/20 0.35
CA14 Q9ULX7 1/20 0.35
IRAK1 P51617 1/20 0.34
MEN1 O00255 2/20 0.33
KMT2A Q03164 2/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
PTGDR2 Q9Y5Y4 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11079176 0.80 CA1 (0.37) IRAK4KDM4EALDH1A1MAPTTHRB
SCHEMBL10649367 0.80 KDM4E (0.36) IRAK4KDM4EALDH1A1MAPTTHRB
SCHEMBL8895550 0.79 MEN1 (0.34) IRAK4KDM4EALDH1A1MAPTTHRB
SCHEMBL10860123 0.79 ACE (0.42) KDM4EALDH1A1
SCHEMBL10545523 0.78 CA1 (0.38) IRAK4KDM4EALDH1A1MAPTTHRB
SCHEMBL11293989 0.78 IRAK4 (0.36) IRAK4KDM4EALDH1A1MAPTTHRB
SCHEMBL11470502 0.76 SDCBP (0.35) IRAK4KDM4EALDH1A1MAPTTHRB
Pyridine SCHEMBL10680880 0.73 ALDH1A1 (0.34) IRAK4KDM4EALDH1A1MAPTTHRB
SCHEMBL11414269 0.73 KMT2A (0.43) KDM4EALDH1A1MAPTTHRBHSD17B10
SCHEMBL11415414 0.73 ACE (0.35) IRAK4KDM4EALDH1A1MAPTTHRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0123442-B1 IMPROVEMENTS IN OR RELATING TO A PROCESS FOR PRODUCING BETA-LACTAM COMPOUNDS THE UNIVERSITY OF NOTRE DAME DU LAC (US) 1988-06-15 EP disclosed
US-4675399-A N-HYDROXY-2-AZETIDINONES; ACYLATION, SOLVOLYSIS NOTRE DAME UNIVERSITY (US) 1987-06-23 US disclosed
US-4565654-A BETA-LACTAMASE ENZYME INHIBITORS UNIVERSITY OF NOTRE DAME DU LAC (US) 1986-01-21 US disclosed
EP-0123442-A1 Improvements in or relating to a process for producing beta-lactam compounds THE UNIVERSITY OF NOTRE DAME DU LAC (US) 1984-10-31 EP disclosed