SCHEMBL11080306

SCHEMBL11080306

Cc1cc(-c2ccncc2)c(C(C)C)[nH]c1=O

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE3B Q13370 11/20 0.48
PDE3A Q14432 11/20 0.48
AURKB Q96GD4 1/20 0.48
INCENP Q9NQS7 1/20 0.48
CDK5 Q00535 2/20 0.45
CDK5R1 Q15078 2/20 0.45
KDM4E B2RXH2 2/20 0.44
PDE5A O76074 1/20 0.44
LMNA P02545 1/20 0.44
HPGD P15428 1/20 0.44
TSHR P16473 1/20 0.44
PTGS1 P23219 1/20 0.44
PDE4A P27815 1/20 0.44
CYP2C19 P33261 1/20 0.44
BLM P54132 1/20 0.44
PDE4B Q07343 1/20 0.44
PDE4C Q08493 1/20 0.44
PDE4D Q08499 1/20 0.44
CDC7 O00311 1/20 0.43
GSK3B P49841 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11241034 0.83 PDE3B (0.66) PDE3BPDE3AAURKBINCENPCDK5
SCHEMBL11236260 0.83 PDE3B (0.43) PDE3BPDE3AAURKBINCENPCDK5
SCHEMBL11251979 0.81 PDE3B (0.42) PDE3BPDE3AAURKBINCENPCDK5
SCHEMBL11076607 0.80 PDE3B (0.71) PDE3BPDE3AAURKBINCENPKDM4E
SCHEMBL11231010 0.80 PDE3A (0.68) PDE3BPDE3AAURKBINCENPCDK5
SCHEMBL11238710 0.80 CDK5 (0.49) PDE3BPDE3AAURKBINCENPCDK5
SCHEMBL11246267 0.79 PDE3B (0.40) PDE3BPDE3AAURKBINCENPCDK5
SCHEMBL11246751 0.79 CDC7 (0.61) PDE3BPDE3AAURKBINCENPCDK5
SCHEMBL11223807 0.76 CDK5 (0.44) PDE3BPDE3AAURKBINCENPCDK5
SCHEMBL8334066 0.76 CDK5 (0.68) CDK5CDK5R1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0109628-A1 2(1H)-pyridinones and preparation, useful as cardiotonics STERLING DRUG INC. (US) 1984-05-30 EP disclosed