SCHEMBL11246751

SCHEMBL11246751

CC(C)c1[nH]c(=O)c(C(N)=O)cc1-c1ccncc1

nearest known ligand 0.61

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CDC7 O00311 8/20 0.61
CDK5 Q00535 7/20 0.48
CDK5R1 Q15078 7/20 0.48
CCNC P24863 2/20 0.48
CDK8 P49336 2/20 0.48
BTK Q06187 1/20 0.44
PDE3B Q13370 1/20 0.43
PDE3A Q14432 1/20 0.43
AURKB Q96GD4 1/20 0.43
INCENP Q9NQS7 1/20 0.43
IKBKB O14920 1/20 0.42
CHUK O15111 1/20 0.42
IKBKE Q14164 1/20 0.42
PKMYT1 Q99640 1/20 0.42
CCNA2 P20248 1/20 0.42
CDK2 P24941 1/20 0.42
CCNA1 P78396 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11238710 0.88 CDK5 (0.49) CDC7CDK5CDK5R1CCNCCDK8
SCHEMBL11223811 0.86 CDC7 (0.48) CDC7CDK5CDK5R1CCNCCDK8
SCHEMBL11242338 0.83 CDK5 (0.51) CDC7CDK5CDK5R1PDE3BPDE3A
SCHEMBL10704473 0.82 CCNC (0.67) CDC7CDK5CDK5R1CCNCCDK8
SCHEMBL11223807 0.82 CDK5 (0.44) CDC7CDK5CDK5R1CCNCCDK8
SCHEMBL11231253 0.81 CDC7 (0.48) CDC7CCNCCDK8BTKPDE3B
SCHEMBL11241034 0.80 PDE3B (0.66) CDC7CDK5CDK5R1CCNCCDK8
SCHEMBL8334162 0.79 CDK5 (0.74) CDC7CDK5CDK5R1
SCHEMBL11080306 0.79 PDE3B (0.48) CDC7CDK5CDK5R1CCNCCDK8
SCHEMBL11239860 0.78 CDC7 (0.48) CDC7CCNCCDK8BTKPDE3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4365065-A 1-(Pyridinyl)-2-(dimethylamino)ethenyl lower-alkyl ketones STERLING DRUG INC. (US) 1982-12-21 US disclosed
US-4313951-A 3-Substituted-6-(lower-alkyl)-5-(pyridinyl)-2(1H)-pyridinones, their cardiotonic use and intermediates therefor STERLING DRUG INC. (US) 1982-02-02 US disclosed