SCHEMBL11080446

SCHEMBL11080446

CCOc1ccc(C2CN=C(N)N(C)C2)cc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
MAPT P10636 3/20 0.40
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
NQO1 P15559 1/20 0.39
CTSD P07339 1/20 0.38
BACE1 P56817 1/20 0.38
BACE2 Q9Y5Z0 1/20 0.38
ALDH1A1 P00352 2/20 0.37
ACACB O00763 2/20 0.37
POLB P06746 1/20 0.37
TP53 P04637 1/20 0.37
HPGD P15428 1/20 0.37
HTT P42858 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
LMNA P02545 1/20 0.37
MAOA P21397 1/20 0.36
MAOB P27338 1/20 0.36
GAA P10253 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11079433 0.89 ALDH1A1 (0.40) TSHRMAPTALDH1A1ACACBTP53
SCHEMBL11081528 0.89 HRH3 (0.41) CTSDBACE1BACE2ALDH1A1LMNA
SCHEMBL11080492 0.84 TP53 (0.43) TSHRMAPTBACE1ALDH1A1TP53
SCHEMBL11079297 0.84 ADRA1A (0.43) TDP1KMT2AALDH1A1L3MBTL1MAOA
SCHEMBL11075393 0.81 BRD4 (0.37) TSHRMAPTMEN1KMT2AALDH1A1
SCHEMBL11087497 0.79 BRD4 (0.38) ALDH1A1HTT
SCHEMBL11090881 0.78 SRD5A1 (0.53) TSHRLMNA
SCHEMBL11111651 0.78 BRD4 (0.55) MAOB
SCHEMBL11076487 0.78 BRD4 (0.37) MAOAMAOB
SCHEMBL11080957 0.78 BRD4 (0.37)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0024776-B1 4-PHENYL AND 5-PHENYL-1,4,5,6-TETRAHYDROPYRIMIDINE DERIVATIVES, PHARMACEUTICAL COMPOSITIONS CONTAINING SAID DERIVATIVES, AND PROCESS FOR PREPARING SAID DERIVATIVES SYNTEX (U.S.A.) INC. (US) 1984-12-27 EP disclosed
EP-0024776-A1 4-Phenyl and 5-phenyl-1,4,5,6-tetrahydropyrimidine derivatives, pharmaceutical compositions containing said derivatives, and process for preparing said derivatives SYNTEX (U.S.A.) INC. (US) 1981-03-11 EP disclosed