SCHEMBL11080801

SCHEMBL11080801

O=c1cc2c(n[nH]1)CCNC2

nearest known ligand 0.58

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.58
CYP3A4 P08684 1/20 0.40
HTR2C P28335 1/20 0.37
PNMT P11086 7/20 0.35
CD44 P16070 1/20 0.35
MAOB P27338 1/20 0.35
ADRA2A P08913 2/20 0.34
ADRA2B P18089 2/20 0.34
ADRA2C P18825 2/20 0.34
ASIC3 Q9UHC3 1/20 0.34
PDE4B Q07343 1/20 0.34
PDE3A Q14432 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31130652 0.85 GAA (0.58) GAAHTR2CPNMTCD44MAOB
SCHEMBL27901543 0.82 GAA (0.53) GAAPDE4BPDE3A
Hydrochloric Acid SCHEMBL31233767 0.81 GAA (0.52) GAAPDE4BPDE3A
SCHEMBL20092675 0.75 GAA (0.89) GAAPDE4BPDE3A
SCHEMBL3617104 0.69 GAA (0.56) GAAPDE4BPDE3A
SCHEMBL1875764 0.68
Hydrochloric Acid SCHEMBL30144072 0.67 PNMT (0.39) CYP3A4HTR2CPNMTCD44MAOB
Hydrochloric Acid SCHEMBL31284488 0.67 PNMT (0.39) CYP3A4HTR2CPNMTCD44MAOB
SCHEMBL31126172 0.67 HTR2C (0.79) CYP3A4HTR2CASIC3
SCHEMBL14719247 0.66 PARP1 (0.48) PNMTCD44MAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4478837-A HYPOTENSIVE AGENTS SANDOZ LTD. (CH) 1984-10-23 US disclosed
US-3954754-A ANTIHYPERTENSIVES SANDOZ LTD. (CH) 1976-05-04 US disclosed