SCHEMBL11081129

SCHEMBL11081129

COc1ccc(-c2nc3c4ccc(Cl)cc4ccc3n2C)cc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 1/20 0.48
GABRA2 P47869 1/20 0.42
GABRB2 P47870 1/20 0.42
CYP3A4 P08684 2/20 0.41
TP53 P04637 1/20 0.40
AURKA O14965 1/20 0.40
AURKB Q96GD4 1/20 0.40
GLA P06280 1/20 0.40
ALDH1A1 P00352 1/20 0.40
HPGD P15428 1/20 0.40
EGFR P00533 2/20 0.39
MEN1 O00255 1/20 0.39
MAPT P10636 1/20 0.39
RAB9A P51151 1/20 0.39
KMT2A Q03164 1/20 0.39
ADORA3 P0DMS8 1/20 0.38
ADORA1 P30542 1/20 0.38
CA1 P00915 1/20 0.38
CA2 P00918 1/20 0.38
MAOB P27338 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL11086416 0.88 PARP1 (0.51) PARP1CYP3A4ALDH1A1HPGDMEN1
SCHEMBL11078271 0.87 PARP1 (0.50) PARP1CYP3A4TP53ALDH1A1HPGD
SCHEMBL11075495 0.84 TLR7 (0.50) GABRA2GABRB2EGFRMAPTRAB9A
SCHEMBL11078229 0.84 PARP1 (0.47) PARP1ALDH1A1HPGDMEN1MAPT
SCHEMBL11080557 0.83 PARP1 (0.46) PARP1TP53MAPTDHFRSHMT2
SCHEMBL11086406 0.83 PARP1 (0.46) PARP1ALDH1A1HPGDMEN1MAPT
SCHEMBL11080835 0.83 PARP1 (0.46) PARP1GABRA2GABRB2TP53ALDH1A1
SCHEMBL11076059 0.82 TLR7 (0.48) PARP1TP53ALDH1A1HPGDMEN1
SCHEMBL11083854 0.82 PARP1 (0.46) PARP1ADORA3ADORA1DHFRSHMT2
SCHEMBL11073129 0.82 PARP1 (0.55) PARP1TP53ALDH1A1HPGDMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4435417-A ANTIINFLAMMATORY AGENTS GRUPPO LEPETIT S.P.A. (IT) 1984-03-06 US disclosed
EP-0012866-A1 New 3H-naphtho(1,2-d)imidazoles, processes for preparing them, compounds for use as antiinflammatory and antimicrobial agents and compositions for that use containing them GRUPPO LEPETIT S.P.A. (IT) 1980-07-09 EP disclosed