SCHEMBL11084405

SCHEMBL11084405

Cc1c(C(=O)O)c(CC(=O)O)n(C)c1C(=O)c1cccn1C

nearest known ligand 0.37

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.36
HSD17B10 Q99714 1/20 0.36
NPC1 O15118 2/20 0.36
RAB9A P51151 2/20 0.36
PKM P14618 1/20 0.35
NFKB1 P19838 1/20 0.35
NFKB2 Q00653 1/20 0.35
RELA Q04206 1/20 0.35
MAOB P27338 1/20 0.35
CXCL8 P10145 1/20 0.34
AKR1B1 P15121 1/20 0.34
PTGS1 P23219 1/20 0.34
PTGS2 P35354 1/20 0.34
GLO1 Q04760 1/20 0.34
TP53 P04637 1/20 0.33
PTGDR2 Q9Y5Y4 1/20 0.33
CYP2C9 P11712 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11091595 0.87 SMN1; SMN2 (0.40) SMN1; SMN2HSD17B10NPC1RAB9A
SCHEMBL7681255 0.77 PTGS2 (0.51) SMN1; SMN2NPC1RAB9ACXCL8AKR1B1
SCHEMBL11087572 0.77 KMT2A (0.42) SMN1; SMN2NPC1RAB9A
SCHEMBL10912428 0.75 PTGS2 (0.42) SMN1; SMN2HSD17B10NPC1RAB9ACXCL8
SCHEMBL7675435 0.75 PTGS2 (0.57) SMN1; SMN2CXCL8AKR1B1PTGS1PTGS2
SCHEMBL11088533 0.74 PTGS2 (0.59) SMN1; SMN2HSD17B10NPC1RAB9APKM
SCHEMBL11198226 0.73 PTGS2 (0.33) CXCL8AKR1B1PTGS1PTGS2GLO1
SCHEMBL10881482 0.68 PTGS2 (0.41) SMN1; SMN2HSD17B10NPC1RAB9ANFKB1
SCHEMBL526662 0.68 SMN1; SMN2 (0.58) SMN1; SMN2HSD17B10NPC1RAB9APKM
SCHEMBL11087575 0.68 USP2 (0.41) SMN1; SMN2NPC1RAB9ACYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4434175-A 5-AROYL-PYRROLE ALKANOIC ACIDS MERCK & CO., INC. (US) 1984-02-28 US disclosed
EP-0072013-A1 Pyrrole compounds as anti-inflammatory and analgesic agents MERCK & CO. INC. (US) 1983-02-16 EP disclosed