SCHEMBL11084408

SCHEMBL11084408

CSC1=Nc2ccccc2C(c2ccccc2)=NC1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 1/20 0.49
GABRA1 P14867 4/20 0.43
GABRG2 P18507 4/20 0.43
GABRB3 P28472 4/20 0.43
GABRA5 P31644 4/20 0.43
GABRA3 P34903 4/20 0.43
GABRA2 P47869 4/20 0.43
GABRB2 P47870 4/20 0.43
CCKBR P32239 1/20 0.43
CHRM1 P11229 2/20 0.43
CCNB2 O95067 1/20 0.37
CDK1 P06493 1/20 0.37
CCNB1 P14635 1/20 0.37
GSK3B P49841 1/20 0.37
CCNB3 Q8WWL7 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
OPRK1 P41145 2/20 0.35
GABRP O00591 1/20 0.35
GABRD O14764 1/20 0.35
CACNA1F O60840 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11086081 0.83 OPRK1 (0.50) GABRA1GABRG2GABRB3GABRA5GABRA3
SCHEMBL11834281 0.81 GABRA1 (0.40) GABRA1GABRG2GABRB3GABRA5GABRA3
SCHEMBL10469905 0.77 IDO1 (0.51) IDO1GABRA1GABRG2GABRB3GABRA5
SCHEMBL28297205 0.77 IDO1 (0.51) IDO1GABRA1GABRG2GABRB3GABRA5
SCHEMBL7312843 0.76 IDO1 (0.47) IDO1GABRA1GABRG2GABRB3GABRA5
SCHEMBL11382448 0.73 IDO1 (0.47) IDO1GABRA1GABRG2GABRB3GABRA5
SCHEMBL10965471 0.73 IDO1 (0.47) IDO1GABRA1GABRG2GABRB3GABRA5
SCHEMBL27926926 0.73 IDO1 (0.47) IDO1GABRA1GABRG2GABRB3GABRA5
SCHEMBL18977949 0.72 IDO1 (0.69) IDO1GSK3BL3MBTL1LMNAGAA
SCHEMBL7307922 0.72 IDO1 (0.43) IDO1GABRA1GABRG2GABRB3GABRA5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4427590-A Triazolobenzodiazepine derivatives CIBA-GEIGY CORPORATION (US) 1984-01-24 US disclosed
US-4017492-A As-triazinobenzodiazepin-1-ones THE UPJOHN COMPANY (US) 1977-04-12 US disclosed
US-3946032-A Acetal derivatives of 6-phenyl-4H-s-triazolo[4,3-a][1,4]benzodiazepine-1-carboxaldehyde CIBA-GEIGY CORPORATION (US) 1976-03-23 US disclosed