SCHEMBL11085549

SCHEMBL11085549

CC(C(=O)O)c1ccc2nc3cc(C(F)(F)F)c(Cl)cn3c(=O)c2c1

nearest known ligand 0.46

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 11/20 0.46
AKR1C2 P52895 11/20 0.46
PTAFR P25105 5/20 0.38
ALPG P10696 1/20 0.38
TBXAS1 P24557 3/20 0.37
CHRM1 P11229 1/20 0.37
PTGS1 P23219 1/20 0.37
AKR1C4 P17516 1/20 0.36
AKR1C1 Q04828 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11082982 0.85 AKR1C3 (0.44) AKR1C3AKR1C2PTAFRALPGTBXAS1
SCHEMBL11079315 0.82 AKR1C3 (0.45) AKR1C3AKR1C2PTAFRALPGTBXAS1
SCHEMBL11090785 0.80 KDM4E (0.48) PTAFRALPGTBXAS1
SCHEMBL11084425 0.78 ALPG (0.46) PTAFRALPGTBXAS1
SCHEMBL11083819 0.77 ALPG (0.47) PTAFRALPGTBXAS1
SCHEMBL11085352 0.76 ALPG (0.40) PTAFRALPGTBXAS1
SCHEMBL11089935 0.76 ALPG (0.46) PTAFRALPGTBXAS1
SCHEMBL11082635 0.76 MAOA (0.41) AKR1C3AKR1C2CHRM1PTGS1
SCHEMBL11259134 0.76 KDM4E (0.53) PTAFRALPGTBXAS1PTGS1
SCHEMBL11076242 0.76 ALPG (0.64) PTAFRALPGTBXAS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4457927-A Pyrido[2,1-b]quinazolinone derivatives and the preparation and use thereof SCHERING, AKTIENGESELLSCHAFT (DE) 1984-07-03 US disclosed