SCHEMBL11086808

SCHEMBL11086808

COc1ccc(CC2N(C)CCC(=O)C2(C)C)cc1

nearest known ligand 0.48

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
GLA P06280 1/20 0.47
NPSR1 Q6W5P4 1/20 0.47
HSD11B1 P28845 2/20 0.46
BCHE P06276 1/20 0.45
ACHE P22303 1/20 0.45
GAA P10253 1/20 0.45
SIGMAR1 Q99720 1/20 0.43
PTGS1 P23219 1/20 0.42
PTGS2 P35354 1/20 0.42
POLB P06746 2/20 0.41
HRH3 Q9Y5N1 1/20 0.41
TLR9 Q9NR96 1/20 0.41
CMA1 P23946 1/20 0.41
MEN1 O00255 1/20 0.40
TSHR P16473 1/20 0.40
KMT2A Q03164 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL11082477 0.99 GLA (0.46) GLANPSR1HSD11B1BCHEACHE
SCHEMBL11733135 0.83 SIGMAR1 (0.50) GAASIGMAR1MEN1KMT2A
Hydrochloric Acid SCHEMBL11731711 0.82 SIGMAR1 (0.49) GAASIGMAR1MEN1KMT2A
Hydrochloric Acid SCHEMBL11731633 0.81 GAA (0.40) GAAHRH3MEN1KMT2A
SCHEMBL11730460 0.74 SIGMAR1 (0.43) GLANPSR1BCHEACHESIGMAR1
SCHEMBL31013097 0.73 GLA (0.46) GLANPSR1GAATLR9MEN1
SCHEMBL11084149 0.73 BCHE (0.44) GLANPSR1BCHEACHEGAA
SCHEMBL11085223 0.73 SIGMAR1 (0.42) GLANPSR1BCHEACHESIGMAR1
SCHEMBL3009582 0.73 GLA (0.46) GLANPSR1GAATLR9MEN1
SCHEMBL11731603 0.73 GLA (0.40) GLANPSR1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0028717-B1 6,7-BENZOMORPHAN DERIVATIVES, PROCESSES FOR THEIR PRODUCTION, PHARMACEUTICAL COMPOSITIONS CONTAINING SAID DERIVATIVES AND THEIR USE AS PHARMACEUTICALS ACF CHEMIEFARMA NV (NL) 1984-08-15 EP disclosed
US-4425353-A Analgesic 5-oxygenated-6,7-benzomorphan derivatives ACF CHEMIEFARMA NV (NL) 1984-01-10 US disclosed
US-4406904-A Method of inhibiting luteinizing hormone secretion with 6,7-benzomorphan derivatives ACF CHEMIEFARMA NV (NL) 1983-09-27 US disclosed
EP-0028717-A1 6,7-Benzomorphan derivatives, processes for their production, pharmaceutical compositions containing said derivatives and their use as pharmaceuticals ACF CHEMIEFARMA NV (NL) 1981-05-20 EP disclosed
US-4012392-A ANALGESICS, MORPHINE ANTAGONISTS ACF CHEMIEFARMA N.V. (NL) 1977-03-15 US disclosed