SCHEMBL11087707

SCHEMBL11087707

COc1ccc(C([C]=O)OCc2ccccc2)cc1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AOC3 Q16853 1/20 0.55
CA1 P00915 1/20 0.50
CA2 P00918 1/20 0.50
ACHE P22303 1/20 0.50
CNR2 P34972 1/20 0.48
LTA4H P09960 1/20 0.47
ALDH1A1 P00352 2/20 0.46
HTT P42858 1/20 0.45
TSHR P16473 1/20 0.45
NPC1 O15118 2/20 0.44
RAB9A P51151 1/20 0.44
ACP3 P15309 1/20 0.44
L3MBTL1 Q9Y468 2/20 0.43
PBRM1 Q86U86 1/20 0.43
PPARG P37231 1/20 0.43
PPARA Q07869 1/20 0.43
FFAR1 O14842 2/20 0.43
ATM Q13315 1/20 0.43
POLB P06746 1/20 0.42
TDP1 Q9NUW8 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2673956 0.85 SLC6A2 (0.45) CA1CA2ALDH1A1HTTTSHR
SCHEMBL11106772 0.80 AOC3 (0.60) AOC3CA1CA2ACHECNR2
SCHEMBL5122883 0.77 CNR2 (0.54) AOC3CA1CA2ACHECNR2
SCHEMBL28451883 0.77 AOC3 (0.53) AOC3CA1CA2ACHECNR2
SCHEMBL11754330 0.76 ALDH1A1 (0.54) CNR2LTA4HALDH1A1TSHRACP3
SCHEMBL11324514 0.75 ATM (0.46) AOC3LTA4HALDH1A1ACP3PBRM1
SCHEMBL10964256 0.75 AOC3 (0.54) AOC3CA1CA2ACHECNR2
SCHEMBL10964251 0.75 CNR2 (0.51) AOC3CA1CA2ACHECNR2
SCHEMBL3932308 0.73 LTA4H (0.58) AOC3LTA4HNPC1L3MBTL1FFAR1
SCHEMBL15514667 0.73 LTA4H (0.53) AOC3LTA4HALDH1A1HTTNPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4461726-A Desulfurization of penicillins to prepare azetidinones HOFFMANN-LA ROCHE INC. (US) 1984-07-24 US disclosed
US-4195021-A 1,3-Disubstituted 2-azetidinone antibitotics ELI LILLY AND COMPANY (US) 1980-03-25 US disclosed
EP-0001715-A2 Azetidinone antibiotics and their pharmaceutical formulations and use ELI LILLY AND COMPANY (US) 1979-05-02 EP disclosed