SCHEMBL11090108

SCHEMBL11090108

CS(=O)(=O)c1ccc(-c2[nH]c(C(N)(C(F)(F)F)C(F)(F)F)nc2-c2ccccc2)cc1

nearest known ligand 0.62

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PTGS1 P23219 10/20 0.62
PTGS2 P35354 10/20 0.62
ALDH1A1 P00352 2/20 0.51
HPGD P15428 1/20 0.51
ESR1 P03372 1/20 0.50
ESR2 Q92731 1/20 0.50
ALOX5 P09917 1/20 0.46
CSNK1A1 P48729 1/20 0.46
CSNK1D P48730 1/20 0.46
CSNK1E P49674 1/20 0.46
MAPK11 Q15759 1/20 0.46
MAPK14 Q16539 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
CSNK1A1L Q8N752 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11087266 0.91 PTGS2 (0.64) PTGS1PTGS2ALDH1A1ALOX5CSNK1A1
SCHEMBL7488369 0.91 PTGS2 (0.64) PTGS1PTGS2ALDH1A1ALOX5CSNK1A1
SCHEMBL7084859 0.88 PTGS2 (0.67) PTGS1PTGS2ALDH1A1HPGDESR1
SCHEMBL10878849 0.86 PTGS1 (0.62) PTGS1PTGS2ALDH1A1HPGDESR1
SCHEMBL7088151 0.84 PTGS1 (0.69) PTGS1PTGS2ALDH1A1HPGD
SCHEMBL11083668 0.81 ESR1 (0.52) PTGS1PTGS2ALDH1A1HPGDESR1
SCHEMBL10852756 0.80 PTGS2 (0.41) PTGS1PTGS2ALDH1A1ALOX5CSNK1A1
SCHEMBL11087907 0.78 ESR1 (0.47) ALDH1A1HPGDESR1ESR2CSNK1A1
SCHEMBL7084237 0.78 PTGS2 (0.55) PTGS1PTGS2ALDH1A1ESR1ESR2
SCHEMBL213705 0.78 PTGS2 (0.70) PTGS1PTGS2ALDH1A1ESR1ESR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4472422-A Antihypertensive 4,5-diaryl-α-polyfluoro-alkyl-1H-imidazole-2-methanamines E. I. DU PONT DE NEMOURS AND COMPANY (US) 1984-09-18 US claimed
US-4472422-A Antihypertensive 4,5-diaryl-α-polyfluoro-alkyl-1H-imidazole-2-methanamines E. I. DU PONT DE NEMOURS AND COMPANY (US) 1984-09-18 US disclosed