SCHEMBL11092102

SCHEMBL11092102

CCCCCNC1(c2ccc(O)cc2)CCC(=O)CC1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRIN2D O15399 2/20 0.36
GRIN3B O60391 2/20 0.36
GRIA1 P42261 2/20 0.36
GRIA2 P42262 2/20 0.36
GRIA3 P42263 2/20 0.36
GRIA4 P48058 2/20 0.36
GRIN1 Q05586 2/20 0.36
GRIN2A Q12879 2/20 0.36
GRIN2B Q13224 2/20 0.36
GRIN2C Q14957 2/20 0.36
GRIN3A Q8TCU5 2/20 0.36
HSD17B3 P37058 7/20 0.36
NAAA Q02083 1/20 0.35
ESR1 P03372 3/20 0.35
ADRA2A P08913 2/20 0.35
ADORA3 P0DMS8 2/20 0.35
TACR2 P21452 2/20 0.35
SLC6A2 P23975 2/20 0.35
SLC6A4 P31645 2/20 0.35
SLC6A3 Q01959 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11089351 0.84 DRD3 (0.43)
SCHEMBL11093324 0.83 DRD3 (0.45) GRIN2DGRIN3BGRIA1GRIA2GRIA3
SCHEMBL11094533 0.80 DRD3 (0.41) SLC6A4
Ethylene SCHEMBL11093778 0.78 DRD3 (0.40) SLC6A4
SCHEMBL19095278 0.75 MEN1 (0.49) GRIN2DGRIN3BGRIA1GRIA2GRIA3
SCHEMBL11557919 0.74 DRD3 (0.38) SLC6A4CHRM2ACHE
SCHEMBL11097718 0.73 ALDH1A1 (0.37) HSD17B10ALDH1A1LMNACYP3A4PTGS2
Hydrochloric Acid SCHEMBL11099779 0.73 ALDH1A1 (0.37) HSD17B10ALDH1A1LMNACYP3A4
SCHEMBL11096000 0.72 GRIN2D (0.48) GRIN2DGRIN3BGRIA1GRIA2GRIA3
SCHEMBL11095882 0.72 EPHX1 (0.34)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4460604-A ANALGESICS, NARCOTIC ANTAGONIST THE UPJOHN COMPANY (US) 1984-07-17 US claimed
US-4460604-A ANALGESICS, NARCOTIC ANTAGONIST THE UPJOHN COMPANY (US) 1984-07-17 US disclosed
US-4180584-A ANALGESIC; NARCOTIC ANTAGONIST THE UPJOHN COMPANY (US) 1979-12-25 US disclosed
US-4065573-A ANALGESICS THE UPJOHN COMPANY (US) 1977-12-27 US disclosed