SCHEMBL11093050

SCHEMBL11093050

N#CC1(c2ccc(Cl)cc2Cl)CCC(=O)CC1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A3 Q01959 5/20 0.39
SLC6A4 P31645 4/20 0.39
PDE4A P27815 1/20 0.36
PDE4B Q07343 1/20 0.36
PDE4C Q08493 1/20 0.36
PDE4D Q08499 1/20 0.36
ALDH1A1 P00352 1/20 0.35
OPRM1 P35372 2/20 0.35
PSEN1 P49768 1/20 0.35
PSEN2 P49810 1/20 0.35
APH1B Q8WW43 1/20 0.35
NCSTN Q92542 1/20 0.35
APH1A Q96BI3 1/20 0.35
PSENEN Q9NZ42 1/20 0.35
GABRA1 P14867 3/20 0.34
GABRG2 P18507 3/20 0.34
GABRB3 P28472 3/20 0.34
GABRB1 P18505 2/20 0.34
GABRB2 P47870 2/20 0.34
OTUD7B Q6GQQ9 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL838201 0.87 SLC6A4 (0.45) SLC6A3SLC6A4ALDH1A1OPRM1GABRA1
SCHEMBL29457607 0.87 SLC6A4 (0.45) SLC6A3SLC6A4ALDH1A1OPRM1GABRA1
SCHEMBL17543073 0.86 PSEN1 (0.42) PDE4APDE4BPDE4CPDE4DOPRM1
SCHEMBL11468178 0.83 SLC6A4 (0.50) SLC6A3SLC6A4ALDH1A1OPRM1PDE7A
SCHEMBL18742609 0.83 SLC6A4 (0.46) SLC6A3SLC6A4ALDH1A1OPRM1GABRA1
SCHEMBL8184370 0.82 SLC6A4 (0.53) SLC6A3SLC6A4ALDH1A1OPRM1PDE7A
SCHEMBL2288498 0.81 ADRA1A (0.42) SLC6A4PDE4APDE4BPDE4CPDE4D
SCHEMBL28678474 0.79 SLC6A4 (0.40) SLC6A3SLC6A4ALDH1A1OPRM1SLC6A2
SCHEMBL6962020 0.79 HTR2C (0.40) SLC6A3SLC6A4ALDH1A1OPRM1SLC6A2
SCHEMBL11119613 0.79 PDE4A (0.51) PDE4APDE4BPDE4CPDE4DALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4460604-A ANALGESICS, NARCOTIC ANTAGONIST THE UPJOHN COMPANY (US) 1984-07-17 US disclosed
US-4180584-A ANALGESIC; NARCOTIC ANTAGONIST THE UPJOHN COMPANY (US) 1979-12-25 US disclosed
US-4065573-A ANALGESICS THE UPJOHN COMPANY (US) 1977-12-27 US disclosed