SCHEMBL11096060

SCHEMBL11096060

Cc1c(N)c(C(=O)c2ccccc2)cc(Cl)c1Cl

nearest known ligand 0.51

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CHRM4 P08173 1/20 0.47
MAPT P10636 3/20 0.46
GAA P10253 1/20 0.46
ALOX15 P16050 2/20 0.45
POLB P06746 2/20 0.44
MAPK14 Q16539 2/20 0.44
MAPK13 O15264 1/20 0.44
MAPK12 P53778 1/20 0.44
MAPK11 Q15759 1/20 0.44
ALDH1A1 P00352 3/20 0.43
LMNA P02545 2/20 0.43
MEN1 O00255 1/20 0.41
USP2 O75604 1/20 0.41
GLA P06280 1/20 0.41
KMT2A Q03164 1/20 0.41
HSD17B10 Q99714 1/20 0.41
PBRM1 Q86U86 1/20 0.41
ADORA1 P30542 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15792781 0.85 MAPT (0.50) MAPTGAAALOX15POLBMAPK14
SCHEMBL27566029 0.82 MAPT (0.50) MAPTGAAALOX15POLBMAPK14
SCHEMBL951003 0.80 KDM4E (0.48) MAPTGAAALDH1A1MEN1KMT2A
SCHEMBL11519197 0.79 AKR1C3 (0.44) MAPTGAAALOX15POLBALDH1A1
SCHEMBL27585830 0.79 MAPT (0.50) CHRM4MAPTGAAPOLBMAPK14
SCHEMBL28747892 0.79 MAPT (0.50) MAPTGAAALOX15POLBMAPK14
SCHEMBL19253323 0.78 MAPT (0.53) MAPTGAAALOX15POLBMAPK14
SCHEMBL28404725 0.77 AKR1C3 (0.46) CHRM4MAPTGAAALOX15MAPK14
SCHEMBL11215128 0.76 MAPT (0.60) MAPTGAAALOX15POLBMAPK14
SCHEMBL5079583 0.76 AKR1C3 (0.48) MAPTGAAALOX15POLBMAPK14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0044091-B1 PROCESS FOR THE PREPARATION OF N-ALKYLAMINO-BENZOPHENONES PIERRE FABRE S.A. (FR) 1984-01-11 EP disclosed
EP-0010030-B1 DERIVATIVES OF 2'-(ORTHO-CHLORO-BENZOYL),4'-CHLORO-GLYCIN ANILIDE, THEIR PREPARATION AND THEIR USE IN MEDICINES PIERRE FABRE S.A. (FR) 1982-05-05 EP disclosed
EP-0044091-A2 Process for the preparation of N-alkylamino-benzophenones PIERRE FABRE S.A. (FR) 1982-01-20 EP disclosed