SCHEMBL11097294

SCHEMBL11097294

c1ccc(C(=NCc2cccc(CN=C(c3ccccc3)c3ccccc3)c2)c2ccccc2)cc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRIN2B Q13224 9/20 0.54
GRIN1 Q05586 4/20 0.53
GRIN2D O15399 2/20 0.53
GRIN3B O60391 2/20 0.53
GRIN2A Q12879 2/20 0.53
GRIN2C Q14957 2/20 0.53
GRIN3A Q8TCU5 2/20 0.53
NOS2 P35228 3/20 0.46
NOS1 P29475 3/20 0.46
ALDH1A1 P00352 2/20 0.46
NOS3 P29474 2/20 0.46
SMN1; SMN2 Q16637 2/20 0.46
CYP3A4 P08684 1/20 0.46
NFKB1 P19838 1/20 0.46
HTR3E A5X5Y0 1/20 0.44
HTR3B O95264 1/20 0.44
HTR3A P46098 1/20 0.44
HTR3D Q70Z44 1/20 0.44
HTR3C Q8WXA8 1/20 0.44
HTR1A P08908 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5075641 0.89 GRIN2B (0.63) GRIN2BGRIN1GRIN2DGRIN3BGRIN2A
SCHEMBL6495653 0.89 GRIN2B (0.49) GRIN2BGRIN1GRIN2DGRIN3BGRIN2A
SCHEMBL11094429 0.85 GRIN2B (0.57) GRIN2BGRIN1GRIN2DGRIN3BGRIN2A
SCHEMBL19745518 0.83 GRIN2B (0.61) GRIN2BGRIN1MEN1KMT2A
SCHEMBL30389572 0.81 GRIN2B (0.53) GRIN2BGRIN1CYP1A2MEN1KMT2A
SCHEMBL14587410 0.80 GRIN2B (0.44) GRIN2BGRIN1HTR3EHTR3BHTR3A
SCHEMBL8544952 0.79 GRIN2B (0.67) GRIN2BGRIN1NOS2RAB9A
SCHEMBL8548012 0.79 SCN2A (0.55) GRIN2BGRIN1NOS2ALDH1A1RAB9A
SCHEMBL10692194 0.78 GRIN2B (0.50) GRIN2BGRIN1SMN1; SMN2RAB9AMEN1
SCHEMBL7076954 0.76 GRIN2B (0.59) GRIN2BGRIN1NOS2SMN1; SMN2KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4448776-A Method of using certain substituted aliphatic secondary amines or their salts for easing breathing BUCHER KARL (CH) 1984-05-15 US disclosed
EP-0058373-A1 Substituted aliphatic secondary amines and their salts, pharmaceutical compositions containing them and their use CIBA-GEIGY AG (CH) 1982-08-25 EP disclosed