SCHEMBL11099522

SCHEMBL11099522

C[C@@H](Nc1nc2ccccc2o1)C(=O)O

nearest known ligand 0.54

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 5/20 0.54
RAB9A P51151 5/20 0.54
GAA P10253 2/20 0.54
SMN1; SMN2 Q16637 4/20 0.51
ALDH1A1 P00352 3/20 0.51
PKM P14618 3/20 0.51
NPSR1 Q6W5P4 1/20 0.51
SCD O00767 1/20 0.51
ELANE P08246 4/20 0.51
TP53 P04637 2/20 0.49
LMNA P02545 2/20 0.46
USP2 O75604 1/20 0.46
HSD17B10 Q99714 1/20 0.46
ALOX15 P16050 1/20 0.46
MAPT P10636 1/20 0.46
CSNK1D P48730 1/20 0.45
HSP90AA1 P07900 1/20 0.44
PCSK9 Q8NBP7 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16972933 1.00 NPC1 (0.54) NPC1RAB9AGAASMN1; SMN2ALDH1A1
SCHEMBL16972931 1.00 NPC1 (0.54) NPC1RAB9AGAASMN1; SMN2ALDH1A1
SCHEMBL13127921 0.88 NPC1 (0.50) NPC1RAB9AGAASMN1; SMN2ALDH1A1
SCHEMBL22561750 0.87 NPC1 (0.49) NPC1RAB9AGAASMN1; SMN2ALDH1A1
SCHEMBL2543164 0.85 ELANE (0.55) NPC1RAB9AGAASMN1; SMN2ALDH1A1
SCHEMBL2541599 0.85 NPC1 (0.51) NPC1RAB9AGAASMN1; SMN2ALDH1A1
SCHEMBL11269418 0.84 ALDH1A1 (0.46) NPC1RAB9AGAAALDH1A1ELANE
SCHEMBL4464723 0.81 NPC1 (0.52) NPC1RAB9AGAASMN1; SMN2ALDH1A1
SCHEMBL11100838 0.81 RAB9A (0.51) NPC1RAB9AGAASMN1; SMN2ALDH1A1
SCHEMBL3953148 0.80 ELANE (0.61) NPC1RAB9AGAASMN1; SMN2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0042753-B1 NONAPEPTIDE AND DECAPEPTIDE AGONISTS OF LUTEINIZING HORMONE RELEASING HORMONE CONTAINING HETEROCYCLIC AMINO ACID RESIDUES, METHODS FOR THEIR PREPARATION, PHARMACEUTICAL COMPOUNDS CONTAINING THEM, AND THEIR PHARMACEUTICAL USE SYNTEX (U.S.A.) INC. (US) 1984-03-21 EP disclosed
US-4318905-A Nonapeptide and decapeptide agonists of luteinizing hormone releasing hormone containing heterocyclic amino acid residues SYNTEX (U.S.A.) INC. (US) 1982-03-09 US disclosed
EP-0042753-A1 Nonapeptide and decapeptide agonists of luteinizing hormone releasing hormone containing heterocyclic amino acid residues, methods for their preparation, pharmaceutical compounds containing them, and their pharmaceutical use SYNTEX (U.S.A.) INC. (US) 1981-12-30 EP disclosed