SCHEMBL11099951

SCHEMBL11099951

COc1ccc(C(O)CNCc2ccccc2)cc1OC

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRB2 P07550 6/20 0.61
OPRK1 P41145 1/20 0.55
ADRB1 P08588 3/20 0.53
LMNA P02545 2/20 0.53
ALDH1A1 P00352 1/20 0.53
NPSR1 Q6W5P4 1/20 0.53
SLC22A1 O15245 1/20 0.53
CHRM2 P08172 1/20 0.53
CYP3A4 P08684 1/20 0.53
CHRM1 P11229 1/20 0.53
TSHR P16473 1/20 0.53
NFKB1 P19838 1/20 0.53
SLC6A4 P31645 1/20 0.53
OPRM1 P35372 1/20 0.53
SLC6A3 Q01959 1/20 0.53
HIF1A Q16665 1/20 0.53
ADRB3 P13945 3/20 0.53
MEN1 O00255 1/20 0.52
KMT2A Q03164 1/20 0.52
DRD2 P14416 4/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17527284 0.91 BCHE (0.55) ADRB2OPRK1ADRB1LMNAMEN1
SCHEMBL8906047 0.88 ADRB3 (0.60) ADRB2OPRK1ADRB1LMNAALDH1A1
SCHEMBL8906311 0.88 ADRB2 (0.55) ADRB2OPRK1ADRB1LMNAALDH1A1
SCHEMBL8904588 0.87 OPRK1 (0.57) ADRB2OPRK1ADRB1LMNAALDH1A1
SCHEMBL8904970 0.87 OPRK1 (0.57) ADRB2OPRK1ADRB1LMNAALDH1A1
SCHEMBL9590684 0.86 ADRB2 (0.76) ADRB2OPRK1ADRB1LMNAALDH1A1
SCHEMBL8907024 0.86 OPRK1 (0.56) ADRB2OPRK1ADRB1LMNAALDH1A1
SCHEMBL11102216 0.85 MEN1 (0.59) ADRB2OPRK1ADRB1LMNAALDH1A1
SCHEMBL23022855 0.84 BCHE (0.52) ADRB2LMNAALDH1A1HIF1AMEN1
SCHEMBL1438054 0.84 BCHE (0.55) ADRB2OPRK1DRD2DRD1DRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0040956-B1 8-SUBSTITUTED 4-(3,4-DIHYDROXYPHENYL)-1,2,3,4-TETRAHYDROISOQUINOLINES SMITHKLINE BECKMAN CORPORATION (US) 1984-10-31 EP disclosed
US-4340600-A Renal dilating methods and compositions using 4-(3,4-dihydroxyphenyl)-1,2,3,4-tetrahydroisoquinolines SMITHKLINE CORPORATION (US) 1982-07-20 US disclosed
EP-0040956-A1 8-Substituted 4-(3,4-dihydroxyphenyl)-1,2,3,4-tetrahydroisoquinolines SMITHKLINE BECKMAN CORPORATION (US) 1981-12-02 EP disclosed