SCHEMBL11110139

SCHEMBL11110139

CC1=C(C(=O)OCCC#N)C(c2ccccc2F)C(C(=O)OC(C)C)=C(C)N1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR3C2 P08235 3/20 0.48
CACNA1C Q13936 4/20 0.46
ACHE P22303 1/20 0.46
CYP3A4 P08684 5/20 0.46
CYP2C9 P11712 5/20 0.46
CYP2C19 P33261 5/20 0.46
CYP1A2 P05177 4/20 0.46
MEN1 O00255 3/20 0.46
KMT2A Q03164 3/20 0.46
LMNA P02545 2/20 0.46
CYP2D6 P10635 2/20 0.46
TSHR P16473 1/20 0.46
NFKB1 P19838 1/20 0.46
THPO P40225 1/20 0.46
MAPT P10636 1/20 0.46
CACNA1F O60840 2/20 0.44
CACNA1D Q01668 2/20 0.44
CACNA1S Q13698 2/20 0.44
HTT P42858 1/20 0.43
MLNR O43193 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6950267 0.87 CYP1A2 (0.58) CACNA1CACHECYP3A4CYP2C9CYP2C19
SCHEMBL10988598 0.87 CACNA1F (0.61) CACNA1CCACNA1FCACNA1DCACNA1S
SCHEMBL8091053 0.82 NR3C2 (0.48) NR3C2CACNA1CCYP3A4CYP2C9CYP2C19
SCHEMBL11276232 0.82 TSHR (0.39) NR3C2CACNA1CACHECYP3A4CYP2C9
SCHEMBL10695488 0.81 CACNA1C (0.61) NR3C2CACNA1CACHECYP3A4CYP2C9
SCHEMBL11376558 0.81 NR3C2 (0.52) NR3C2CACNA1CCYP3A4CYP2C9CYP2C19
SCHEMBL11102848 0.81 KDM4E (0.62) NR3C2CACNA1CCYP3A4CYP2C9CYP2C19
SCHEMBL10748814 0.80 CYP1A2 (0.72) NR3C2CACNA1CCYP3A4CYP2C9CYP2C19
SCHEMBL11131329 0.80 CACNA1C (0.44) NR3C2CACNA1CCYP3A4CYP2C9CYP2C19
SCHEMBL8790137 0.80 TBXA2R (0.49) CACNA1CCYP3A4CYP2C9CYP2C19CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4483985-A ALKALINE HYDROLYSIS OF ESTER GROUP BAYER AKTIENGESELLSCHAFT (DE) 1984-11-20 US disclosed
US-4285955-A CARDIOTONIC, HYPOTENSIVE, AND ANTISPASMOTIC AGENTS; VASODILATION BAYER AKTIENGESELLSCHAFT (DE) 1981-08-25 US disclosed