SCHEMBL11276232

SCHEMBL11276232

CC1=C(OC(=O)OCCC#N)C(c2ccccc2F)C(OC(=O)OC(C)C)=C(C)N1

nearest known ligand 0.46

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
TSHR P16473 3/20 0.39
ALDH1A1 P00352 3/20 0.39
CYP3A4 P08684 2/20 0.39
CYP2C9 P11712 2/20 0.39
CYP2C19 P33261 2/20 0.39
CYP1A2 P05177 1/20 0.39
HSD17B10 Q99714 1/20 0.39
NR3C2 P08235 3/20 0.37
ACHE P22303 1/20 0.36
ALOX15 P16050 1/20 0.35
GAA P10253 2/20 0.34
HTT P42858 1/20 0.34
CACNA1C Q13936 2/20 0.33
CACNA1F O60840 1/20 0.33
CACNA1D Q01668 1/20 0.33
CACNA1S Q13698 1/20 0.33
KDM4E B2RXH2 1/20 0.33
THRB P10828 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11110139 0.82 NR3C2 (0.48) TSHRCYP3A4CYP2C9CYP2C19CYP1A2
SCHEMBL11500369 0.82 NR3C2 (0.46) TSHRALDH1A1CYP3A4CYP2C9CYP2C19
SCHEMBL11291512 0.82 KDM4E (0.47) ALDH1A1CYP2C9CYP2C19HSD17B10NR3C2
SCHEMBL10913788 0.81 CACNA1C (0.54) TSHRALDH1A1CYP3A4CYP2C9CYP2C19
SCHEMBL11498937 0.80 POLB (0.44) TSHRALDH1A1HSD17B10ALOX15GAA
SCHEMBL11500155 0.80 ALDH1A1 (0.44) TSHRALDH1A1CYP3A4CYP2C9CYP2C19
SCHEMBL8949402 0.80 CACNA1D (0.41) TSHRALDH1A1CYP3A4CYP2C9CYP2C19
SCHEMBL11291917 0.80 CACNA1F (0.52) TSHRCYP3A4CYP2C9CYP2C19CYP1A2
SCHEMBL11281855 0.79 KDM4E (0.44) TSHRALDH1A1HSD17B10ALOX15GAA
SCHEMBL11280776 0.79 CACNA1B (0.44) TSHRCYP3A4CYP2C9CYP2C19CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0011706-B1 PROCESS FOR THE PREPARATION OF DERIVATIVES OF 1,4-DIHYDROPYRIDINE-3-CARBOXYLIC ACID, DERIVATIVES OF 1,4-DIHYDROPYRIDINE-3-CARBOXYLIC ACID AND THE USE OF THESE DERIVATIVES FOR THE PREPARATION OF 1,4-DIHYDROPYRIDINE-3,5-DICARBOXYLATES BAYER AG (DE) 1982-03-03 EP disclosed
EP-0011706-A1 Process for the preparation of derivatives of 1,4-dihydropyridine-3-carboxylic acid, derivatives of 1,4-dihydropyridine-3-carboxylic acid and the use of these derivatives for the preparation of 1,4-dihydropyridine-3,5-dicarboxylates BAYER AG (DE) 1980-06-11 EP disclosed