SCHEMBL1111154

SCHEMBL1111154

CC(=O)NC(C)Cc1cccc(C(F)(F)F)n1

nearest known ligand 0.49

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
ACACB O00763 14/20 0.49
P2RX7 Q99572 1/20 0.44
ADAMTS4 O75173 1/20 0.41
MMP13 P45452 1/20 0.41
ADRB1 P08588 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8186745 0.77 IDH1 (0.43) P2RX7ADAMTS4MMP13ADRB1
SCHEMBL1118071 0.77 ACACB (0.43) ACACB
SCHEMBL4664170 0.77 NPSR1 (0.70) P2RX7ADAMTS4MMP13ADRB1NPSR1
SCHEMBL29676316 0.75 ACACB (0.53) ACACBP2RX7ADRB1NPSR1
SCHEMBL1111196 0.74 HTR2A (0.47) P2RX7ADAMTS4MMP13ADRB1
SCHEMBL26046016 0.74 P2RX7 (0.49) P2RX7ADAMTS4MMP13ADRB1NPSR1
Hydrochloric Acid SCHEMBL1111187 0.73 HTR2A (0.46) P2RX7ADAMTS4MMP13ADRB1
SCHEMBL19837388 0.73 P2RX7 (0.47) ACACBP2RX7ADAMTS4MMP13ADRB1
SCHEMBL8256625 0.73 P2RX7 (0.41) P2RX7ADAMTS4MMP13ADRB1
SCHEMBL3823658 0.72 ACACB (0.52) ACACB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2278968-A2 1,5-DIPHENYL-PYRROLIDIN-2-ONE COMPOUNDS AS CB-1 LIGANDS ELI LILLY AND COMPANY (US) 2011-02-02 EP disclosed
WO-2009131814-A2 1,5-DIPHENYL-PYRROLIDIN-2-ONE COMPOUNDS AS CB-1 LIGANDS ELI LILLY AND COMPANY (US) 2009-10-29 WO disclosed