SCHEMBL1111229

SCHEMBL1111229

CC(C)(C)C1COC(c2ccccc2P(c2ccccc2)c2ccccc2)=N1

nearest known ligand 0.35

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
DRD1 P21728 2/20 0.35
MAPT P10636 2/20 0.34
NPC1 O15118 1/20 0.34
RAB9A P51151 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
CNR2 P34972 1/20 0.32
POLB P06746 1/20 0.32
P2RY1 P47900 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15478440 1.00 DRD1 (0.35) DRD1MAPTNPC1RAB9ASMN1; SMN2
SCHEMBL30220116 1.00 DRD1 (0.35) DRD1MAPTNPC1RAB9ASMN1; SMN2
SCHEMBL1111225 1.00 DRD1 (0.35) DRD1MAPTNPC1RAB9ASMN1; SMN2
SCHEMBL29528319 1.00 DRD1 (0.35) DRD1MAPTNPC1RAB9ASMN1; SMN2
SCHEMBL14498419 0.91 SMN1; SMN2 (0.32) MAPTNPC1RAB9ASMN1; SMN2CNR2
SCHEMBL14498430 0.90 NPC1 (0.32) MAPTNPC1RAB9ASMN1; SMN2CNR2
SCHEMBL14498409 0.90 DRD1 (0.33) DRD1MAPTNPC1RAB9ASMN1; SMN2
SCHEMBL23119029 0.88 P2RY1 (0.31) MAPTNPC1RAB9ASMN1; SMN2P2RY1
SCHEMBL14523590 0.88 P2RY1 (0.31) MAPTNPC1RAB9ASMN1; SMN2P2RY1
SCHEMBL14498394 0.87 DRD1 (0.33) DRD1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 86 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113651863-B Unsaturated thioglycoside compound and selective synthesis method and application thereof 华东师范大学 2023-11-10 CN claimed
CN-115677580-A Tetrahydroquinoline spiro alkaloid containing quaternary carbon indandione, preparation method thereof and application thereof in preparing antitumor drugs 中南民族大学 2023-02-03 CN claimed
CN-109721508-B Method for preparing 3-pentenenitrile 安徽省安庆市曙光化工股份有限公司 2022-10-04 CN claimed
CN-113651863-A Unsaturated thioglycoside compound and selective synthesis method and application thereof 华东师范大学 2021-11-16 CN claimed
CN-109721508-A A method of preparing 3 pentene nitrile 安徽省安庆市曙光化工股份有限公司 2019-05-07 CN claimed
CN-109651195-A The method of 2- allyl acetonitrile isomerization reaction generation 3 pentene nitrile 安徽省安庆市曙光化工股份有限公司 2019-04-19 CN claimed
EP-2443128-B1 New synthetic route for the preparation of alpha-amino boronic esters LEK PHARMACEUTICALS (SI) 2017-12-20 EP claimed
EP-2443129-B1 PROCESS FOR HYDROGENATION OF HALOGENOALKENES WITHOUT DEHALOGENATION LEK PHARMACEUTICALS (SI) 2016-11-23 EP claimed
US-9315525-B2 Synthetic route for the preparation of α-amino boronic acid derivatives via substituted alk-1-ynes LEK PHARMACEUTICALS D.D. (SI) 2016-04-19 US claimed
US-8785674-B2 Process for hydrogenation of halogenoalkenes without dehalogenation LEK PHARMACEUTICALS D.D. (SL) 2014-07-22 US claimed
US-20120231993-A1 NEW SYNTHETIC ROUTE FOR THE PREPARATION OF ALPHA-AMINO BORONIC ACID DERIVATIVES via SUBSTITUTED ALK-1-YNES LEK PHARMACEUTICALS D.D. (SI) 2012-09-13 US claimed
US-20120220794-A1 PROCESS FOR HYDROGENATION OF HALOGENOALKENES WITHOUT DEHALOGENATION LEK PHARMACEUTICALS D.D. (SI) 2012-08-30 US claimed
EP-2443128-A2 New synthetic route for the preparation of alpha-amino boronic esters LEK Pharmaceuticals d.d. (SI) 2012-04-25 EP claimed
EP-2443129-A2 PROCESS FOR HYDROGENATION OF HALOGENOALKENES WITHOUT DEHALOGENATION LEK Pharmaceuticals d.d. (SI) 2012-04-25 EP claimed
EP-2280016-A1 New synthetic route for the preparation of alpha-amino boronic esters via substituted alk-1-ynes LEK Pharmaceuticals d.d. (SI) 2011-02-02 EP claimed
WO-2010146176-A2 PROCESS FOR HYDROGENATION OF HALOGENOALKENES WITHOUT DEHALOGENATION LEK PHARMACEUTICALS D.D. (SI) 2010-12-23 WO claimed
WO-2010146172-A2 NEW SYNTHETIC ROUTE FOR THE PREPARATION OF α-AMINO BORONIC ACID DERIVATIVES VIA SUBSTITUTED ALK-1-YNES LEK PHARMACEUTICALS D.D. (SI) 2010-12-23 WO claimed
CN-116444400-A Chiral alpha- (trichloromethyl) amine compound and preparation method thereof 合肥工业大学 2023-07-18 CN disclosed
US-20060084820-A1 Enantioselective, catalytic allylation of ketones and olefins CALIFORNIA INSTITUTE OF TECHNOLOGY (US) 2006-04-20 US disclosed
US-6551467-B1 Microwave heated very rapid highly selective (chemo-, regio-and stereo-) allylic substitutions utilising molybdenum or palladium together with an auxiliary ligand as catalytic system PERSONAL CHEMISTRY I UPPSALA AB (SE) 2003-04-22 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060084820-A1 Enantioselective, catalytic allylation of ketones and olefins AKR1C2, TECR, AKR1C4 DRD1 2207/4885MAPT 2756/4885NPC1 1539/4885
US-20120220794-A1 PROCESS FOR HYDROGENATION OF HALOGENOALKENES WITHOUT DEHALOGENATION HDHD5, DEK, HCK DRD1 557/4885MAPT 3500/4885NPC1 3437/4885
US-20120231993-A1 NEW SYNTHETIC ROUTE FOR THE PREPARATION OF ALPHA-AMINO BORONIC ACID DERIVATIVES via SUBSTITUTED ALK-1-YNES ALK, ABL2, ALKBH3 DRD1 559/4885MAPT 2338/4885NPC1 2759/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.