SCHEMBL11113361

SCHEMBL11113361

COc1ccc2c(c1)C(NC1CN3CCC1CC3)c1ccccc1CO2

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRNA7 P36544 4/20 0.44
HTR3A P46098 3/20 0.44
DRD2 P14416 2/20 0.40
DRD3 P35462 2/20 0.40
KDM4E B2RXH2 1/20 0.39
NPC1 O15118 1/20 0.39
ALDH1A1 P00352 1/20 0.39
GAA P10253 1/20 0.39
MAPT P10636 1/20 0.39
HPGD P15428 1/20 0.39
ALOX12 P18054 1/20 0.39
RAB9A P51151 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
CHRM2 P08172 1/20 0.38
CHRM1 P11229 1/20 0.38
CHRM3 P20309 1/20 0.38
DRD1 P21728 2/20 0.37
DRD4 P21917 1/20 0.36
DRD5 P21918 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11109479 0.86 CHRNA7 (0.41) CHRNA7HTR3ACHRM2CHRM1CHRM3
SCHEMBL11128579 0.84 CHRM3 (0.42) CHRNA7HTR3ADRD2DRD3CHRM2
SCHEMBL11117209 0.84 HTR3A (0.41) CHRNA7HTR3ADRD2DRD3GAA
SCHEMBL11116121 0.83 CHRM3 (0.38) CHRNA7HTR3AALDH1A1CHRM2CHRM1
SCHEMBL11113541 0.83 CHRM2 (0.38) CHRNA7GAASMN1; SMN2CHRM2CHRM1
SCHEMBL11115203 0.83 CHRM2 (0.39) CHRNA7HTR3ACHRM2CHRM1CHRM3
SCHEMBL11115200 0.80 CHRNA7 (0.38) CHRNA7HTR3ACHRM2CHRM1CHRM3
SCHEMBL11111944 0.80 CHRM2 (0.36) CHRNA7HTR3AALDH1A1GAAMAPT
SCHEMBL11115518 0.80 CHRM2 (0.36) CHRNA7ALDH1A1GAACHRM2CHRM1
SCHEMBL11000923 0.80 CHRM2 (0.43) CHRNA7CHRM2CHRM1CHRM3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0038564-B1 DIBENZ (B,E) OXEPIN DERIVATIVES AND PHARMACEUTICAL COMPOSITIONS COMPRISING THEM KYOWA HAKKO KOGYO CO., LTD (JP) 1984-09-12 EP disclosed
US-4396550-A ANTICHOLINERGIC, ANTIHISTIMINIC AGENTS KYOWA HAKKO KOGYO CO., LTD. (JP) 1983-08-02 US disclosed
EP-0038564-A1 Dibenz (b,e) oxepin derivatives and pharmaceutical compositions comprising them KYOWA HAKKO KOGYO CO., LTD (JP) 1981-10-28 EP disclosed