SCHEMBL11114047

SCHEMBL11114047

O=C(Nc1ccc(-c2ccc(=O)[nH]n2)cc1)SCc1cccc(C(F)(F)F)c1

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AURKB Q96GD4 3/20 0.67
NTRK1 P04629 2/20 0.67
NTRK2 Q16620 2/20 0.67
JAK2 O60674 1/20 0.67
RET P07949 1/20 0.67
PDGFRB P09619 1/20 0.67
CDK8 P49336 1/20 0.67
NTRK3 Q16288 1/20 0.67
KDR P35968 4/20 0.50
AKR1B1 P15121 2/20 0.47
L3MBTL1 Q9Y468 3/20 0.43
MAPT P10636 3/20 0.43
HPGD P15428 2/20 0.43
NPSR1 Q6W5P4 2/20 0.43
ALDH1A1 P00352 2/20 0.43
CYP1A2 P05177 1/20 0.42
CYP3A4 P08684 1/20 0.42
ALPG P10696 1/20 0.42
CYP2C9 P11712 1/20 0.42
CYP2C19 P33261 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11118397 0.83 AURKB (0.70) AURKBNTRK1NTRK2JAK2RET
SCHEMBL11120834 0.82 AURKB (0.67) AURKBNTRK1NTRK2JAK2RET
SCHEMBL11114055 0.80 KMT2A (0.49) AURKBNTRK1NTRK2JAK2RET
SCHEMBL11116147 0.79 JAK2 (0.55) AURKBNTRK1NTRK2JAK2RET
SCHEMBL11119913 0.78 KDR (0.48) AURKBNTRK1NTRK2JAK2RET
SCHEMBL11116148 0.78 LMNA (0.57) AURKBNTRK1NTRK2JAK2RET
SCHEMBL11119210 0.77 CYP1A2 (0.50) AURKBNTRK1NTRK2JAK2RET
SCHEMBL11119091 0.77 NTRK1 (0.70) AURKBNTRK1NTRK2JAK2RET
SCHEMBL11119331 0.76 LMNA (0.60) AURKBNTRK1NTRK2JAK2RET
SCHEMBL11121541 0.75 JAK2 (0.50) AURKBNTRK1NTRK2JAK2RET

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0116853-A1 Pyridazinones, processes for preparing them, therapeutical compositions containing these compounds and their use BASF Aktiengesellschaft (DE) 1984-08-29 EP disclosed