SCHEMBL11114824

SCHEMBL11114824

Cc1ccc(S(=O)(=O)N2CCC(C(=O)O)(c3cccc(C(F)(F)F)c3)CC2)cc1

nearest known ligand 0.71

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CYP2C19 P33261 1/20 0.71
KMT2A Q03164 5/20 0.58
MEN1 O00255 4/20 0.57
ALDH1A1 P00352 2/20 0.51
LMNA P02545 2/20 0.49
HSD17B10 Q99714 1/20 0.49
TSHR P16473 2/20 0.48
SMN1; SMN2 Q16637 3/20 0.47
L3MBTL1 Q9Y468 1/20 0.47
MAPT P10636 1/20 0.47
XBP1 P17861 1/20 0.47
HTT P42858 1/20 0.47
MAPK1 P28482 1/20 0.46
POLB P06746 1/20 0.46
TRPV4 Q9HBA0 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11120143 0.91 CYP2C19 (0.57) CYP2C19KMT2AMEN1ALDH1A1LMNA
SCHEMBL11114408 0.87 MEN1 (0.55) CYP2C19KMT2AMEN1ALDH1A1LMNA
SCHEMBL11111683 0.81 MEN1 (0.57) CYP2C19KMT2AMEN1ALDH1A1LMNA
SCHEMBL696251 0.77 AKR1C3 (0.67) KMT2AMEN1MAPTHTT
SCHEMBL5726893 0.77 AKR1C3 (0.54) KMT2AMEN1LMNAPOLB
SCHEMBL8747120 0.75 AKR1C3 (0.60)
SCHEMBL3116411 0.75 AKR1C3 (0.60)
SCHEMBL3214214 0.74 ALDH1A1 (0.71) KMT2AMEN1ALDH1A1LMNAHSD17B10
SCHEMBL2701748 0.74 CHRNA7 (0.49) KMT2AMEN1
SCHEMBL11117181 0.73 CYP2C19 (0.67) CYP2C19KMT2AMEN1ALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0034415-B1 1-(CYCLOHEXYL OR CYCLOHEXENYL)-4-ARYL-4-PIPERIDINECARBOXYLIC ACID DERIVATIVES JANSSEN PHARMACEUTICA N.V. (BE) 1984-05-30 EP disclosed
US-4369184-A ANTIHISTAMINES; HETEROCYCLIC NITRILES JANSSEN PHARMACEUTICA N.V. (BE) 1983-01-18 US disclosed