SCHEMBL11115897

SCHEMBL11115897

NC(=CC(=O)c1ccccc1)c1ccccc1.[NaH]

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NFE2L2 Q16236 1/20 0.59
HDAC1 Q13547 2/20 0.55
HDAC2 Q92769 2/20 0.55
MEN1 O00255 2/20 0.53
KMT2A Q03164 2/20 0.53
ALDH1A1 P00352 6/20 0.52
TDP1 Q9NUW8 2/20 0.52
MAPK1 P28482 1/20 0.52
HDAC3 O15379 1/20 0.52
NCOR2 Q9Y618 1/20 0.52
MAPT P10636 4/20 0.50
RECQL P46063 3/20 0.50
TSHR P16473 2/20 0.50
AKT1 P31749 1/20 0.50
POLB P06746 1/20 0.50
CYP3A4 P08684 1/20 0.50
PARP1 P09874 1/20 0.50
CYP2C19 P33261 1/20 0.50
BLM P54132 1/20 0.50
PMP22 Q01453 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11115893 1.00 NFE2L2 (0.59) NFE2L2HDAC1HDAC2MEN1KMT2A
SCHEMBL29089429 0.98 NFE2L2 (0.61) NFE2L2HDAC1HDAC2MEN1KMT2A
SCHEMBL3140459 0.98 NFE2L2 (0.61) NFE2L2HDAC1HDAC2MEN1KMT2A
SCHEMBL3140451 0.98 NFE2L2 (0.61) NFE2L2HDAC1HDAC2MEN1KMT2A
SCHEMBL29089413 0.90 NFE2L2 (0.53) NFE2L2HDAC1HDAC2MEN1KMT2A
SCHEMBL29089423 0.88 NFE2L2 (0.52) NFE2L2HDAC1HDAC2MEN1KMT2A
SCHEMBL29089431 0.87 POLB (0.55) NFE2L2HDAC1HDAC2MEN1KMT2A
SCHEMBL29089415 0.87 MAPT (0.51) NFE2L2HDAC1HDAC2MEN1KMT2A
SCHEMBL29089436 0.87 CYP1B1 (0.53) NFE2L2HDAC1HDAC2MEN1KMT2A
SCHEMBL29089427 0.87 POLB (0.55) NFE2L2HDAC1HDAC2MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0030351-B1 ERGOLINE DERIVATIVES, THEIR PREPARATION AND THERAPEUTIC COMPOSITION CONTAINING THEM FARMITALIA CARLO ERBA S.p.A. (IT) 1984-08-08 EP disclosed
US-4382940-A ANTIDEPRESSANTS, TRANQUILLIZERS, NEUROLENTIC AGENTS, HORMONE INHIB FARMITALIA CARLO ERBA S.P.A. (IT) 1983-05-10 US disclosed
EP-0030351-A2 Ergoline derivatives, their preparation and therapeutic composition containing them FARMITALIA CARLO ERBA S.p.A. (IT) 1981-06-17 EP disclosed