SCHEMBL11116312

SCHEMBL11116312

CCOC(=O)CCc1ccc(C#N)cc1Cl

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP4F2 P78329 3/20 0.47
CYP4A11 Q02928 3/20 0.47
USP14 P54578 2/20 0.45
PDCD1 Q15116 1/20 0.41
CD274 Q9NZQ7 1/20 0.41
P2RX7 Q99572 1/20 0.41
GPR35 Q9HC97 1/20 0.41
ALDH1A1 P00352 3/20 0.40
FFAR1 O14842 1/20 0.40
FFAR4 Q5NUL3 1/20 0.40
GAA P10253 2/20 0.40
PTPN1 P18031 1/20 0.39
KDM4E B2RXH2 1/20 0.38
GLA P06280 1/20 0.38
MAPT P10636 1/20 0.38
HPGD P15428 1/20 0.38
STAT6 P42226 1/20 0.38
KMT2A Q03164 1/20 0.38
HIF1A Q16665 1/20 0.38
AR P10275 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16110186 0.86 PDCD1 (0.43) USP14PDCD1CD274P2RX7GPR35
SCHEMBL8361251 0.81 CYP4F2 (0.53) CYP4F2CYP4A11ALDH1A1GAAPTPN1
SCHEMBL901696 0.81 CYP4F2 (0.53) CYP4F2CYP4A11ALDH1A1GAAKDM4E
SCHEMBL5990825 0.80 CYP4F2 (0.51) CYP4F2CYP4A11ALDH1A1GAAKDM4E
SCHEMBL11112081 0.80 FFAR1 (0.51) P2RX7ALDH1A1FFAR1FFAR4
SCHEMBL11116918 0.78 CYP3A4 (0.44) PDCD1CD274P2RX7GPR35ALDH1A1
SCHEMBL30353239 0.77 CYP4F2 (0.46) CYP4F2CYP4A11USP14PDCD1CD274
SCHEMBL17922634 0.77 CYP4F2 (0.46) CYP4F2CYP4A11USP14PDCD1CD274
Hydrochloric Acid SCHEMBL6873181 0.77 CYP4F2 (0.40) CYP4F2CYP4A11USP14PDCD1CD274
SCHEMBL6870504 0.77 CYP1A2 (0.41) CYP4F2CYP4A11USP14PDCD1CD274

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0038071-B1 NEW UNLABELLED AND RADIOACTIVE LABELLED DERIVATIVES OF BUTYLAMINO PROPIOPHENONE, THEIR PREPARATION, IMMUNOGENS OBTAINED FROM THE UNLABELLED DERIVATIVES AND A PROCESS FOR IMMUNOGEN PREPARATION, ANTISERA RAISED USING THE IMMUNOGENS AND A METHOD FOR RAISING ANTISERA, A RADIOIMMUNOASSAY METHOD AND A TEST KIT FOR USE IN THE ASSAY METHOD THE WELLCOME FOUNDATION LIMITED (GB) 1984-11-14 EP disclosed
US-4356165-A Bupropion radioimmunoassay, and kit BURROUGHS WELLCOME CO. (US) 1982-10-26 US disclosed
US-4355179-A Radioactive nuclide labeled propiophenone compounds BURROUGHS WELLCOME CO. (US) 1982-10-19 US disclosed
US-4347177-A Compounds and methods of making them BURROUGHS WELLCOME CO. (US) 1982-08-31 US disclosed
US-4347382-A 3H Labeled compounds BURROUGHS WELLCOME CO. (US) 1982-08-31 US disclosed
US-4347176-A Compounds and methods of making same BURROUGHS WELLCOME CO. (US) 1982-08-31 US disclosed
US-4347178-A Compounds and methods of making BURROUGHS WELLCOME CO. (US) 1982-08-31 US disclosed
EP-0038071-A2 New unlabelled and radioactive labelled derivatives of butylamino propiophenone, their preparation, immunogens obtained from the unlabelled derivatives and a process for immunogen preparation, antisera raised using the immunogens and a method for raising antisera, a radioimmunoassay method and a test kit for use in the assay method THE WELLCOME FOUNDATION LIMITED (GB) 1981-10-21 EP disclosed